SCHEMBL7302310

SCHEMBL7302310

CCCC[C@@H](C(=O)OCC)N1CCN[C@H](Cc2ccccc2)C1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA4 P22748 2/20 0.41
CA9 Q16790 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
SLC6A2 P23975 3/20 0.39
SLC6A3 Q01959 3/20 0.39
SLC6A4 P31645 2/20 0.39
CNR2 P34972 1/20 0.37
POLB P06746 1/20 0.36
HDAC1 Q13547 1/20 0.36
ABCB1 P08183 1/20 0.36
ACE P12821 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB3 P13945 1/20 0.35
KCNH2 Q12809 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303601 1.00 CA1 (0.41) CA1CA2CA4CA9L3MBTL1
SCHEMBL7302302 1.00 CA1 (0.41) CA1CA2CA4CA9L3MBTL1
SCHEMBL7296229 0.87 CA1 (0.45) CA1CA2CA4CA9SLC6A2
SCHEMBL7296235 0.87 CA1 (0.45) CA1CA2CA4CA9SLC6A2
SCHEMBL7302308 0.77 SLC6A4 (0.44) CA1CA2CA4CA9L3MBTL1
SCHEMBL14983612 0.74 POLB (0.47) CA1CA2CA4CA9SLC6A2
SCHEMBL14983613 0.74 POLB (0.47) CA1CA2CA4CA9SLC6A2
SCHEMBL13858858 0.74 POLB (0.47) CA1CA2CA4CA9SLC6A2
SCHEMBL9311330 0.72 SLC6A4 (0.52) L3MBTL1SLC6A2SLC6A3SLC6A4ACE
SCHEMBL7346890 0.70 MDM2 (0.40) CNR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164388-A Hypotensive agents, treatment of congestive heart failure ABBOTT LABORATORIES (US) 1992-11-17 US disclosed
EP-0439556-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
WO-1990004917-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1990-05-17 WO disclosed
EP-0365992-A1 Heterocyclic peptide renin inhibitors ABBOTT LABORATORIES (US) 1990-05-02 EP disclosed