Bromide

Bromide

SCHEMBL7303705

C[N+]1(Cc2ccccc2)CCN(c2nc3ccccc3o2)CC1.[Br-]

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.48
MAPT P10636 2/20 0.48
GAA P10253 1/20 0.47
KMT2A Q03164 1/20 0.47
KCNH2 Q12809 1/20 0.46
SORD Q00796 2/20 0.46
HTR1A P08908 1/20 0.44
HTR2C P28335 1/20 0.44
SMN1; SMN2 Q16637 4/20 0.43
HTT P42858 3/20 0.43
NAAA Q02083 1/20 0.43
HCAR2 Q8TDS4 1/20 0.42
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7302309 0.81 GAA (0.46) LMNAMAPTGAAKMT2AKCNH2
Bromide SCHEMBL7307800 0.81 GAA (0.54) LMNAMAPTGAAKMT2AKCNH2
Iodide SCHEMBL7306562 0.80 SORD (0.54) LMNAMAPTGAAKMT2AKCNH2
Iodide SCHEMBL7304073 0.80 SORD (0.52) LMNAMAPTGAAKMT2AKCNH2
Hydrochloric Acid SCHEMBL7305474 0.79 SORD (0.47) LMNAMAPTGAAKMT2AKCNH2
Iodide SCHEMBL7307306 0.79 SORD (0.47) LMNAMAPTGAAKMT2AKCNH2
Iodide SCHEMBL7299396 0.76 SORD (0.50) LMNAMAPTGAAKMT2AKCNH2
Bromide SCHEMBL7304866 0.76 GAA (0.52) LMNAMAPTGAAKMT2AKCNH2
Iodide SCHEMBL7304275 0.75 SORD (0.44) LMNAMAPTGAAKMT2AKCNH2
Iodide SCHEMBL7298086 0.75 SORD (0.48) LMNAMAPTGAAKMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0621271-B1 Benzoxazole derivatives and their use as serotonin 5-HT3 receptor antagonists MEIJI SEIKA KAISHA (JP) 2001-10-17 EP disclosed
US-5631257-A ANTISEROTONIN AGENTS FOR TREATMENT OF NAUSEA AND ANTIEMETICS MEIJI SEIKA KAISHA, LTD. (JP) 1997-05-20 US disclosed
EP-0621271-A1 Benzoxazole derivatives and their use as serotonin 5-HT3 receptor antagonists MEIJI SEIKA KAISHA LTD. (JP) 1994-10-26 EP disclosed