SCHEMBL7304402

SCHEMBL7304402

Cc1cc(C)c2c(c1)CC(CC(=O)C1C(=S)CN[C@@H]1C(=O)N1CCCC1)CC2

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PREP P48147 10/20 0.35
DPP4 P27487 1/20 0.31
FAP Q12884 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7293629 0.87 NR2F2 (0.31)
SCHEMBL7304044 0.83 POLB (0.31)
SCHEMBL7304409 0.82 PREP (0.36) PREPDPP4FAPLMNAMAPT
SCHEMBL7302992 0.82 DPP4 (0.41) PREPDPP4FAP
SCHEMBL7294240 0.81 PREP (0.54) PREP
SCHEMBL7296356 0.81 PREP (0.54) PREP
SCHEMBL7302246 0.81 PREP (0.54) PREP
SCHEMBL7295069 0.79 CYP26A1 (0.42) PREPDPP4
SCHEMBL7303602 0.77 GRIK2 (0.30)
SCHEMBL7292981 0.77 PREP (0.48) PREPDPP4FAPHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017929-A Cholinesterase activator ZERIA PHARMACEUTICAL CO., LTD. (JP) 2000-01-25 US disclosed
EP-0754454-A1 CHOLINESTERASE ACTIVATOR ZERIA PHARMACEUTICAL CO., LTD. (JP) 1997-01-22 EP disclosed
EP-0372484-B1 Condensed benzene derivative ZERIA PHARM CO LTD (JP) 1994-10-26 EP disclosed
US-5028604-A Cognition Activators ZERIA PHARMACEUTICAL CO., LTD. (JP) 1991-07-02 US disclosed
EP-0372484-A2 Condensed benzene derivative ZERIA PHARMACEUTICAL CO., LTD. (JP) 1990-06-13 EP disclosed