SCHEMBL7304930

SCHEMBL7304930

CC(C)=C1C(=O)Nc2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.57
TDO2 P48775 1/20 0.57
TDP1 Q9NUW8 3/20 0.55
MAOA P21397 1/20 0.55
MAOB P27338 1/20 0.55
PDGFRA P16234 1/20 0.55
FER P16591 1/20 0.55
LTK P29376 1/20 0.55
CDK8 P49336 1/20 0.55
ACVR1 Q04771 1/20 0.55
LRRK2 Q5S007 1/20 0.55
DYRK1B Q9Y463 1/20 0.55
MAPT P10636 5/20 0.54
ALDH1A1 P00352 4/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
HTT P42858 3/20 0.54
LMNA P02545 1/20 0.54
TGM2 P21980 1/20 0.54
EPHX2 P34913 1/20 0.53
NPSR1 Q6W5P4 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30681308 1.00 IDO1 (0.57) IDO1TDO2TDP1MAOAMAOB
SCHEMBL12220595 0.85 ACVR1 (0.50) IDO1TDO2TDP1MAOAMAOB
SCHEMBL10399820 0.82 ALDH1A1 (0.53) IDO1TDO2TDP1MAOAMAOB
SCHEMBL1465398 0.82 TDP1 (0.54) IDO1TDO2TDP1MAOAMAOB
SCHEMBL1466156 0.82 TDP1 (0.54) IDO1TDO2TDP1MAOAMAOB
SCHEMBL10399821 0.82 ALDH1A1 (0.53) IDO1TDO2TDP1MAOAMAOB
SCHEMBL11980231 0.80 IDO1 (0.61) IDO1TDO2TDP1MAOAMAOB
SCHEMBL14320160 0.79 IDO1 (0.56) IDO1TDO2TDP1MAOAMAOB
SCHEMBL4165371 0.79 IDO1 (0.56) IDO1TDO2TDP1MAOAMAOB
SCHEMBL4165379 0.79 IDO1 (0.56) IDO1TDO2TDP1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed