SCHEMBL7306064

SCHEMBL7306064

CCc1cc([O])c2c(CC)cccc2c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
CYP2A6 P11509 1/20 0.42
GABRA1 P14867 4/20 0.38
GABRB2 P47870 4/20 0.38
ELANE P08246 6/20 0.36
DAO P14920 1/20 0.36
PARP1 P09874 1/20 0.36
KDM4E B2RXH2 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
TP53 P04637 1/20 0.32
HTR6 P50406 1/20 0.32
MAPT P10636 2/20 0.32
MGLL Q99685 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5248752 0.81 CYP1A2 (0.42) CYP1A2CYP2A6GABRA1GABRB2ELANE
SCHEMBL5248750 0.80 CYP1A2 (0.41) CYP1A2CYP2A6GABRA1GABRB2ELANE
SCHEMBL18244315 0.78 GABRA1 (0.44) CYP1A2GABRA1GABRB2ELANEDAO
SCHEMBL22824269 0.76 CYP1A2 (0.58) CYP1A2CYP2A6PARP1KDM4ETDP1
SCHEMBL18242839 0.73 CYP1A2 (0.50) CYP1A2CYP2A6KDM4ETP53HTR6
SCHEMBL3244580 0.73 GABRA1 (0.52) CYP1A2GABRA1GABRB2ELANEDAO
SCHEMBL24630603 0.72 GABRA1 (0.48) GABRA1GABRB2ELANEDAOKDM4E
SCHEMBL26715141 0.72 ELANE (0.42) CYP1A2CYP2A6GABRA1GABRB2ELANE
SCHEMBL23070782 0.71 CYP1A2 (0.53) CYP1A2CYP2A6GABRA1GABRB2ELANE
SCHEMBL21371241 0.70 CYP1A2 (0.39) CYP1A2CYP2A6GABRA1GABRB2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed