SCHEMBL7306987

SCHEMBL7306987

CCOc1ccc(OCC(=O)O)c2c1C(=O)N(CSc1nnnn1-c1ccccc1)S2(=O)=O

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ELANE P08246 19/20 0.73
ALDH1A1 P00352 1/20 0.50
POLB P06746 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7312086 0.91 ELANE (0.65) ELANEALDH1A1POLBSMN1; SMN2
SCHEMBL7304774 0.90 ELANE (0.75) ELANEALDH1A1POLBSMN1; SMN2
SCHEMBL7315370 0.88 ELANE (0.68) ELANEALDH1A1POLBSMN1; SMN2
SCHEMBL7414358 0.84 ELANE (1.00) ELANEALDH1A1POLBSMN1; SMN2
SCHEMBL7314724 0.80 ELANE (0.66) ELANE
SCHEMBL9314177 0.78 ELANE (0.46) ELANEALDH1A1POLBSMN1; SMN2
SCHEMBL7305964 0.78 ELANE (0.77) ELANEALDH1A1
SCHEMBL7419633 0.75 ELANE (1.00) ELANE
SCHEMBL8479185 0.74 ELANE (0.68) ELANEALDH1A1
SCHEMBL7414675 0.74 ELANE (1.00) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874432-A Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof SANOFI (FR) 1999-02-23 US disclosed
US-5650422-A TREATMENT OF EMPHYSEMA, ARTHRITIS OR PANCREATITIS SANOFI (FR) 1997-07-22 US disclosed
US-5596012-A Saccharin derivatives useful as proteolytic enzyme inhibitors and compositions and method of use thereof STERLING WINTHROP INC. (US) 1997-01-21 US disclosed
US-5236917-A Respiratory system disorders, antiarthritic agents STERLING WINTHROP INC. (US) 1993-08-17 US disclosed
EP-0542372-A1 2-Substituted saccharin derivative proteolytic enzyme inhibitors STERLING WINTHROP INC. (US) 1993-05-19 EP disclosed