SCHEMBL7307333

SCHEMBL7307333

COc1ccc(I)c(CC(=O)Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.49
PTGS1 P23219 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
POLB P06746 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7144108 0.86 HSD17B10 (0.51) HSD17B10PTGS1AKR1C3AKR1C2POLB
SCHEMBL7322443 0.85 HSD17B10 (0.68) HSD17B10PTGS1AKR1C3AKR1C2POLB
SCHEMBL30468420 0.85 HSD17B10 (0.68) HSD17B10PTGS1AKR1C3AKR1C2POLB
SCHEMBL7308036 0.85 HSD17B10 (0.50) HSD17B10PTGS1AKR1C3AKR1C2POLB
SCHEMBL7314138 0.84 POLB (0.48) HSD17B10POLBKDM4ENPC1RAB9A
SCHEMBL10962956 0.82 AKR1C3 (0.52) HSD17B10PTGS1AKR1C3AKR1C2MTNR1A
SCHEMBL16836022 0.81 HSD17B10 (0.50) HSD17B10PTGS1AKR1C3AKR1C2POLB
SCHEMBL892777 0.81 HSD17B10 (0.73) HSD17B10MEN1KMT2AMTNR1AMTNR1B
SCHEMBL8237110 0.81 HSD17B10 (0.50) HSD17B10PTGS1AKR1C3AKR1C2POLB
SCHEMBL30660236 0.81 HSD17B10 (0.73) HSD17B10MEN1KMT2AMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4742084-A Aralykyl (arylethynyl)aralkyl amines and their use as vasodilators and antihypertensives MCNEILAB, INC. (US) 1988-05-03 US disclosed
US-4661635-A ANTIARRHYTHMIA AGENTS MCNEILAB, INC. (US) 1987-04-28 US disclosed
EP-0146271-A2 Aralykyl (arylethynyl) aralkyl amines for use as vasodilators and antihypertensives McNeilab, Inc. (US) 1985-06-26 EP disclosed