SCHEMBL30468420

SCHEMBL30468420

COc1ccc(I)c(CC(=O)O)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.68
AKR1C2 P52895 3/20 0.54
AKR1C3 P42330 3/20 0.54
PTGS1 P23219 2/20 0.54
KDM4E B2RXH2 3/20 0.54
LCK P06239 1/20 0.51
POLB P06746 2/20 0.50
ABL1 P00519 1/20 0.50
MAPT P10636 1/20 0.50
RECQL P46063 1/20 0.50
RIN1 Q13671 1/20 0.50
CTDSP1 Q9GZU7 1/20 0.50
MMP2 P08253 2/20 0.46
MMP12 P39900 2/20 0.46
MMP8 P22894 1/20 0.46
MMP13 P45452 1/20 0.46
MMP14 P50281 1/20 0.46
MMP16 P51512 1/20 0.46
LMNA P02545 1/20 0.44
MMP9 P14780 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7322443 1.00 HSD17B10 (0.68) HSD17B10AKR1C2AKR1C3PTGS1KDM4E
SCHEMBL7144108 0.88 HSD17B10 (0.51) HSD17B10AKR1C2AKR1C3PTGS1KDM4E
SCHEMBL7308036 0.86 HSD17B10 (0.50) HSD17B10AKR1C2AKR1C3PTGS1KDM4E
SCHEMBL7307333 0.85 HSD17B10 (0.49) HSD17B10AKR1C2AKR1C3PTGS1KDM4E
SCHEMBL8589029 0.83 HSD17B10 (0.47) HSD17B10KDM4EPOLBABL1MAPT
SCHEMBL10962956 0.83 AKR1C3 (0.52) HSD17B10AKR1C2AKR1C3PTGS1
SCHEMBL7314187 0.83 POLB (0.65) HSD17B10KDM4EPOLBMAPTLMNA
SCHEMBL10411874 0.82 ALDH1A1 (0.47) HSD17B10AKR1C2AKR1C3PTGS1POLB
SCHEMBL21232836 0.81 PPARG (0.46) HSD17B10KDM4EMAPTLMNAALDH1A1
SCHEMBL15935612 0.81 HSD17B10 (0.70) HSD17B10AKR1C2AKR1C3PTGS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332910-A 2-aminopyrimidine derivatives as kinase inhibitors, preparation and use thereof 江苏威凯尔医药科技有限公司 2023-06-27 CN disclosed