SCHEMBL7307641

SCHEMBL7307641

CCCCc1nc(CO)c(C(N)=O)n1Cc1ccc(-c2ccccc2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.54
AGTR1 P30556 1/20 0.53
AGTR2 P50052 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311709 0.92 AGTR1 (0.54) AGTR1AGTR2
SCHEMBL7301745 0.92 AGTR1 (0.58) AGTR1AGTR2
SCHEMBL7907344 0.91 AGTR1 (0.58) AGTR1AGTR2
SCHEMBL7302138 0.90 AGTR1 (0.51) AGTR1AGTR2
SCHEMBL7308473 0.89 PPARG (0.54) PPARG
SCHEMBL7444657 0.89 AGTR1 (0.55) AGTR1AGTR2
SCHEMBL7307434 0.87 PPARG (0.52) PPARGAGTR1AGTR2
SCHEMBL7300759 0.87 PPARG (0.52) PPARGAGTR1AGTR2
SCHEMBL7314316 0.87 AGTR1 (0.68) AGTR1AGTR2
SCHEMBL7312054 0.87 AGTR1 (0.49) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0545912-B1 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-04-25 EP disclosed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US disclosed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US disclosed
EP-0545912-A2 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1993-06-09 EP disclosed
EP-0503785-A1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1992-09-16 EP disclosed