SCHEMBL7307834

SCHEMBL7307834

Cc1cccc(CNC(=O)N[C@H](C(=O)O)C(C)C)n1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.53
TSHR P16473 1/20 0.53
HSD17B10 Q99714 1/20 0.45
ALDH1A1 P00352 5/20 0.45
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
FPR2 P25090 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307826 1.00 MAPK1 (0.53) MAPK1TSHRHSD17B10ALDH1A1NPSR1
SCHEMBL7800076 0.81 NPSR1 (0.43) MAPK1ALDH1A1NPSR1SMN1; SMN2KEAP1
SCHEMBL6446960 0.80 NPC1 (0.58) MAPK1TSHRALDH1A1POLBSMN1; SMN2
SCHEMBL6446955 0.80 NPC1 (0.58) MAPK1TSHRALDH1A1POLBSMN1; SMN2
SCHEMBL13734815 0.78 NPSR1 (0.59) MAPK1TSHRNPSR1POLBSMN1; SMN2
SCHEMBL7303071 0.78 TYR (0.46) KEAP1NFE2L2
SCHEMBL7308687 0.78 CA2 (0.47) ALDH1A1POLBSMN1; SMN2KEAP1NFE2L2
SCHEMBL7298552 0.78 TYR (0.46) KEAP1NFE2L2
SCHEMBL7308684 0.78 CA2 (0.47) ALDH1A1POLBSMN1; SMN2KEAP1NFE2L2
SCHEMBL5175905 0.76 MAPK1 (0.76) MAPK1TSHRHSD17B10ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed