SCHEMBL7308422

SCHEMBL7308422

C=CC(=O)O[C@H]1[C@H]2C(C)(C)CC[C@H](O[Si](C)(C)C(C)(C)C)[C@]2(C)[C@@]2(O)C(=O)C[C@](C)(C=C)O[C@]2(C)[C@H]1O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADCY1 Q08828 16/20 0.60
MAPK1 P28482 4/20 0.52
CYP3A4 P08684 3/20 0.52
TSHR P16473 2/20 0.52
GMNN O75496 1/20 0.52
BLM P54132 1/20 0.52
PMP22 Q01453 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CYP2D6 P10635 1/20 0.52
NFKB1 P19838 1/20 0.52
HIF1A Q16665 1/20 0.52
NR1I2 O75469 1/20 0.52
CHRM2 P08172 1/20 0.52
ABCB1 P08183 1/20 0.52
HTR1A P08908 1/20 0.52
ADRA2A P08913 1/20 0.52
SLC2A1 P11166 1/20 0.52
HTR2A P28223 1/20 0.52
ADRA1A P35348 1/20 0.52
SCN1A P35498 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10586330 0.93 ADCY1 (0.57) ADCY1MAPK1CYP3A4TSHRGMNN
SCHEMBL10585769 0.93 ADCY1 (0.57) ADCY1MAPK1CYP3A4TSHRGMNN
SCHEMBL10583757 0.90 ADCY1 (0.63) ADCY1MAPK1CYP3A4TSHRGMNN
SCHEMBL7295262 0.89 ADCY1 (0.61) ADCY1MAPK1CYP3A4TSHRNR1I2
SCHEMBL10494966 0.89 ADCY1 (0.58) ADCY1MAPK1CYP3A4TSHRGMNN
SCHEMBL9737018 0.89 ADCY1 (0.58) ADCY1MAPK1CYP3A4TSHRGMNN
SCHEMBL10586036 0.89 ADCY1 (0.53) ADCY1MAPK1CYP3A4TSHRGMNN
SCHEMBL7303938 0.88 ADCY1 (0.54) ADCY1MAPK1CYP3A4TSHRGMNN
SCHEMBL10584713 0.87 ADCY1 (0.52) ADCY1MAPK1CYP3A4TSHRGMNN
SCHEMBL7303390 0.87 ADCY1 (0.53) ADCY1MAPK1CYP3A4TSHRGMNN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0447962-A1 Labdanes and process for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1991-09-25 EP disclosed
EP-0315097-A2 Acyl labdane derivatives, process for their preparation and their use as medicines HOECHST AKTIENGESELLSCHAFT (DE) 1989-05-10 EP disclosed