SCHEMBL7308677

SCHEMBL7308677

CCc1ccc(C(C#N)(CCC=O)C(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 9/20 0.40
CYP3A4 P08684 7/20 0.40
CYP3A5 P20815 1/20 0.40
EBP Q15125 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
ABCC1 P33527 4/20 0.37
TSHR P16473 4/20 0.37
KCNH2 Q12809 3/20 0.37
LMNA P02545 3/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CYP2C19 P33261 2/20 0.37
ABCB11 O95342 2/20 0.37
CACNA1F O60840 2/20 0.37
HTR1A P08908 2/20 0.37
ADRA2A P08913 2/20 0.37
DRD2 P14416 2/20 0.37
ADRA2C P18825 2/20 0.37
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27541310 0.87 ABCB1 (0.39) ABCB1CYP3A4CYP3A5EBPSIGMAR1
SCHEMBL5756895 0.85 EBP (0.39) ABCB1CYP3A4CYP3A5EBPSIGMAR1
SCHEMBL5754384 0.84 EBP (0.38) ABCB1CYP3A4CYP3A5EBPSIGMAR1
SCHEMBL5755590 0.84 EBP (0.38) ABCB1CYP3A4CYP3A5EBPSIGMAR1
SCHEMBL5752959 0.84 EBP (0.51) ABCB1CYP3A4CYP3A5EBPSIGMAR1
SCHEMBL7310593 0.84 EBP (0.51) ABCB1CYP3A4CYP3A5EBPSIGMAR1
SCHEMBL5753427 0.82 CYP3A4 (0.43) ABCB1CYP3A4CYP3A5EBPSIGMAR1
SCHEMBL5751877 0.80 CYP3A4 (0.40) ABCB1CYP3A4CYP3A5TSHRLMNA
SCHEMBL5756697 0.80 EBP (0.35) ABCB1CYP3A4CYP3A5EBPSIGMAR1
SCHEMBL5754191 0.78 CYP3A4 (0.40) ABCB1CYP3A4CYP3A5EBPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed