SCHEMBL7310246

SCHEMBL7310246

O=C(OCc1ccsc1)Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.60
BCL9 O00512 1/20 0.45
CTNNB1 P35222 1/20 0.45
GAA P10253 2/20 0.43
MAOB P27338 1/20 0.41
RAB9A P51151 2/20 0.41
PKM P14618 1/20 0.41
KMT2A Q03164 1/20 0.41
MGLL Q99685 1/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SLC1A3 P43003 2/20 0.40
SLC1A2 P43004 2/20 0.40
SLC1A1 P43005 2/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7365417 0.87 HTR2A (0.49) HTR2ABCL9CTNNB1GAAPKM
SCHEMBL5827968 0.84 HTR2A (0.80) HTR2ABCL9CTNNB1GAAMAOB
SCHEMBL14621621 0.81 HTR2A (0.74) HTR2ABCL9CTNNB1GAAMAOB
SCHEMBL1714950 0.81 HTR2A (0.70) HTR2ABCL9CTNNB1RAB9AKMT2A
SCHEMBL8810198 0.80 CA12 (0.55) MAOB
SCHEMBL23042226 0.78 HTR2A (0.67) HTR2ABCL9CTNNB1GAAMAOB
SCHEMBL6648196 0.78 HTR2A (0.70) HTR2ABCL9CTNNB1GAAMAOB
SCHEMBL6594172 0.78 HTR2A (0.74) HTR2ABCL9CTNNB1GAAMAOB
SCHEMBL4112112 0.78 HTR2A (0.74) HTR2ABCL9CTNNB1GAAMAOB
SCHEMBL20480867 0.78 HTR2A (0.70) HTR2ABCL9CTNNB1GAAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed