SCHEMBL7310575

SCHEMBL7310575

CC(=O)NC1(c2ccccc2)CCN(CCCC(CN(C)C(=O)Cc2ccccc2)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 6/20 0.73
TACR1 P25103 3/20 0.73
CCR5 P51681 1/20 0.61
TACR3 P29371 6/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7750648 0.99 TACR2 (0.72) TACR2TACR1CCR5TACR3
SCHEMBL8972619 0.86 TACR2 (0.60) TACR2TACR1CCR5TACR3
SCHEMBL7311532 0.86 TACR2 (0.72) TACR2TACR1CCR5TACR3
SCHEMBL8971053 0.86 TACR2 (0.60) TACR2TACR1CCR5TACR3
Saredutant SCHEMBL676170 0.84 TACR2 (1.00) TACR2TACR1
Saredutant SCHEMBL29371280 0.84 TACR2 (1.00) TACR2TACR1
Saredutant SCHEMBL185911 0.84 TACR2 (1.00) TACR2TACR1
Saredutant SCHEMBL9317902 0.84 TACR2 (0.98) TACR2TACR1
SCHEMBL7312636 0.83 TACR2 (0.66) TACR2TACR1TACR3
Hydrochloric Acid SCHEMBL7751882 0.82 TACR2 (0.65) TACR2TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673928-A1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists SANOFI (FR) 1995-09-27 EP disclosed