SCHEMBL7311526

SCHEMBL7311526

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(O)CNC[C@@H](O)[C@H](Cc1ccncc1)NC(=O)O

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.55
BACE1 P56817 12/20 0.52
ATM Q13315 1/20 0.52
BCHE P06276 1/20 0.48
PSEN1 P49768 2/20 0.47
PSEN2 P49810 2/20 0.47
APH1B Q8WW43 2/20 0.47
NCSTN Q92542 2/20 0.47
APH1A Q96BI3 2/20 0.47
PSENEN Q9NZ42 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303561 0.93 KLK5 (0.61) KLK5BACE1ATMBCHEPSEN1
SCHEMBL7309398 0.93 KLK5 (0.61) KLK5BACE1ATMBCHEPSEN1
SCHEMBL7309908 0.90 KLK5 (0.65) KLK5BACE1ATMBCHEPSEN1
SCHEMBL13538226 0.88 KLK5 (0.48) KLK5BACE1ATMPSEN1PSEN2
SCHEMBL7311931 0.86 KLK5 (0.54) KLK5BACE1ATMBCHEPSEN1
SCHEMBL7304887 0.86 KLK5 (0.54) KLK5BACE1ATMBCHEPSEN1
SCHEMBL1104912 0.85 KLK5 (0.61) KLK5BACE1ATMBCHEPSEN1
SCHEMBL12103325 0.85 KLK5 (0.61) KLK5BACE1ATMBCHEPSEN1
SCHEMBL8222457 0.85 KLK5 (0.61) KLK5BACE1ATMBCHEPSEN1
SCHEMBL19261937 0.85 KLK5 (0.61) KLK5BACE1ATMBCHEPSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559256-A Aminediol protease inhibitors E. R. SQUIBB & SONS, INC. (US) 1996-09-24 US disclosed
EP-0580402-A2 Aminediol protease inhibitors E.R. SQUIBB & SONS, INC. (US) 1994-01-26 EP disclosed