SCHEMBL7312097

SCHEMBL7312097

C/C(N)=C\C(=O)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
HDAC1 Q13547 2/20 0.55
HDAC2 Q92769 2/20 0.55
ALDH1A1 P00352 4/20 0.52
TDP1 Q9NUW8 2/20 0.52
MAPK1 P28482 2/20 0.52
HDAC3 O15379 1/20 0.52
NCOR2 Q9Y618 1/20 0.52
MAPT P10636 6/20 0.50
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
RECQL P46063 3/20 0.50
GAA P10253 2/20 0.50
POLB P06746 2/20 0.50
HSD17B10 Q99714 2/20 0.50
AKT1 P31749 2/20 0.50
CYP3A4 P08684 2/20 0.50
THRB P10828 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3187174 1.00 NFE2L2 (0.59) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL3187167 1.00 NFE2L2 (0.59) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL11112600 0.98 NFE2L2 (0.57) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL11112598 0.98 NFE2L2 (0.57) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL3875405 0.83 NFE2L2 (0.55) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL3794069 0.83 NFE2L2 (0.55) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL3794074 0.83 NFE2L2 (0.55) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL566675 0.82 NFE2L2 (0.64) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL10984963 0.82 NFE2L2 (0.64) NFE2L2MEN1KMT2AHDAC1HDAC2
SCHEMBL10984957 0.82 NFE2L2 (0.64) NFE2L2MEN1KMT2AHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
EP-0458823-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES. BOEHRINGER MANNHEIM ITALIA (IT) 1991-12-04 EP disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed
EP-0210571-A1 Phosphonopyridines and their 1,4-dihydroderivatives BOEHRINGER BIOCHEMIA ROBIN S.p.A. (IT) 1987-02-04 EP disclosed