SCHEMBL7312299

SCHEMBL7312299

O=C(O)C1CCCCN(S(=O)(=O)c2ccc3ccccc3c2)C1

nearest known ligand 0.93

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 7/20 0.93
AKR1C1 Q04828 3/20 0.84
EIF2AK3 Q9NZJ5 1/20 0.71
MCOLN3 Q8TDD5 3/20 0.63
TSHR P16473 2/20 0.63
MAPT P10636 2/20 0.60
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
LMNA P02545 3/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
ALDH1A1 P00352 2/20 0.54
KDM4E B2RXH2 1/20 0.54
MCL1 Q07820 1/20 0.54
HTT P42858 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246679 0.96 AKR1C3 (1.00) AKR1C3AKR1C1EIF2AK3MCOLN3TSHR
SCHEMBL22191886 0.93 AKR1C3 (1.00) AKR1C3AKR1C1EIF2AK3MCOLN3TSHR
SCHEMBL7303194 0.91 AKR1C3 (1.00) AKR1C3AKR1C1EIF2AK3MCOLN3TSHR
SCHEMBL7304595 0.86 AKR1C3 (0.82) AKR1C3AKR1C1EIF2AK3MCOLN3TSHR
SCHEMBL25269754 0.85 AKR1C3 (0.80) AKR1C3AKR1C1EIF2AK3MCOLN3TSHR
SCHEMBL6791588 0.83 AKR1C3 (0.85) AKR1C3AKR1C1MCOLN3TSHRKMT2A
SCHEMBL5244699 0.83 EIF2AK3 (0.74) AKR1C3AKR1C1EIF2AK3TSHRMEN1
SCHEMBL6079186 0.82 AKR1C3 (0.75) AKR1C3AKR1C1EIF2AK3TSHRMAPT
SCHEMBL4701073 0.82 MAPT (0.77) AKR1C3AKR1C1TSHRMAPTLMNA
SCHEMBL21669903 0.82 MAPT (0.77) AKR1C3AKR1C1TSHRMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0520336-A2 Aldehyde derivatives and their use as calpain inhibitors FUJIREBIO Inc. (JP) 1992-12-30 EP disclosed