SCHEMBL7312903

SCHEMBL7312903

CC(=O)Nc1nc2c(s1)CC(NC(C)=O)CC2

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
GSK3B P49841 2/20 0.51
CSNK2A1 P68400 2/20 0.51
ALDH1A1 P00352 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
HSD17B10 Q99714 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12804717 0.93 GSK3B (0.55) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL1029349 0.93 GSK3B (0.55) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL1030470 0.93 GSK3B (0.55) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL12804931 0.92 NPC1 (0.52) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL3562146 0.92 NPC1 (0.52) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL3562143 0.92 NPC1 (0.52) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL12805601 0.90 TSHR (0.51) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL1073223 0.90 TSHR (0.51) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL3048550 0.90 TSHR (0.51) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1
SCHEMBL7319478 0.89 NPC1 (0.48) NPC1RAB9ASMN1; SMN2GSK3BCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4886812-A REGULATING DOPAMINE CONCENTRATION; PARKINSON DISEASE, HYPOTENSIVE AGENT, SCHIZOPHRENIA DR. KARL THOMAE GMBH (DE) 1989-12-12 US disclosed
US-4843086-A HYPOTENSIVE AGENTS, SCHIZOPHRENIA, PARKINSON'S DISEASE BOEHRINGER INGELHEIM KG (DE) 1989-06-27 US disclosed
US-4731374-A PARKINSON*S DISEASE DR. KARL THOMAE GMBH (DE) 1988-03-15 US disclosed
EP-0186087-A1 Tetrahydro-benzothiazoles, their production and their use as intermediates or drugs Dr. Karl Thomae GmbH (DE) 1986-07-02 EP disclosed