SCHEMBL7313432

SCHEMBL7313432

CON(C)C(=O)[C@H](CSc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 1/20 0.58
BTK Q06187 1/20 0.58
PPARA Q07869 7/20 0.47
PPARG P37231 6/20 0.47
PPARD Q03181 2/20 0.46
MMP13 P45452 1/20 0.45
CTSS P25774 4/20 0.43
CTSK P43235 3/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
ACE P12821 1/20 0.42
MTNR1A P48039 3/20 0.41
MTNR1B P49286 3/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226599 0.88 JAK3 (0.51) JAK3BTKPPARAPPARGPPARD
SCHEMBL7449431 0.85 PPARA (0.67) JAK3BTKPPARAPPARGPPARD
SCHEMBL18549279 0.84 JAK3 (0.56) JAK3BTKPPARAPPARGPPARD
SCHEMBL17028420 0.84 JAK3 (0.56) JAK3BTKPPARAPPARGPPARD
SCHEMBL12617667 0.84 JAK3 (0.56) JAK3BTKPPARAPPARGPPARD
SCHEMBL2951876 0.84 NFKB1 (0.53) PPARAPPARGPPARDMMP13CTSS
SCHEMBL2948733 0.84 NFKB1 (0.53) PPARAPPARGPPARDMMP13CTSS
SCHEMBL4671738 0.84 PPARA (0.64) PPARAPPARGPPARDMMP13CTSS
SCHEMBL5142486 0.84 PPARA (0.64) PPARAPPARGPPARDMMP13CTSS
SCHEMBL4671732 0.84 PPARA (0.64) PPARAPPARGPPARDMMP13CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604183-B1 Inhibitors of HIV protease useful for the treatment of aids LILLY CO ELI (US) 1997-03-05 EP disclosed
US-5514802-A Intermediates for preparing HIV protease inhibitors ELI LILLY AND COMPANY (US) 1996-05-07 US disclosed
US-5475136-A Inhibitors of HIV protease useful for the treatment of AIDS ELI LILLY AND COMPANY (US) 1995-12-12 US disclosed
EP-0604183-A1 Inhibitors of HIV protease useful for the treatment of aids ELI LILLY AND COMPANY (US) 1994-06-29 EP disclosed