SCHEMBL7314514

SCHEMBL7314514

Nc1ccc(C(=O)N2CCc3cn[nH]c3-c3ncccc32)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 9/20 0.46
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
POLB P06746 1/20 0.38
ALOX15 P16050 1/20 0.38
NR4A1 P22736 1/20 0.38
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
GPBAR1 Q8TDU6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8820600 0.86 AVPR2 (0.53) AVPR2LMNASMN1; SMN2NPC1RAB9A
SCHEMBL5236886 0.81 AVPR2 (0.64) AVPR2PDK1PDK2PDK3PDK4
SCHEMBL9059943 0.79 AVPR2 (0.75) AVPR2
SCHEMBL5236665 0.78 AVPR2 (0.58) AVPR2
SCHEMBL5235714 0.74 AVPR2 (0.50) AVPR2GPBAR1
SCHEMBL5235967 0.74 AVPR2 (0.56) AVPR2LMNAPOLB
SCHEMBL5238090 0.73 AVPR2 (0.57) AVPR2LMNASMN1; SMN2RAB9A
SCHEMBL7314107 0.73 HPGD (0.44) AVPR2LMNASMN1; SMN2NPC1RAB9A
SCHEMBL9059936 0.73 AVPR2 (0.46) AVPR2SMN1; SMN2
SCHEMBL8818791 0.72 AVPR2 (0.51) AVPR2LMNASMN1; SMN2NPC1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022295-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed
US-5532235-A TO TREAT EXCESS RENAL REABSORPTION AMERICAN CYANAMID COMPANY (US) 1996-07-02 US disclosed