SCHEMBL7315145

SCHEMBL7315145

COc1c(C(=O)O)cc(Cl)c(N)c1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.46
TPMT P51580 1/20 0.45
ALDH1A1 P00352 5/20 0.44
KDM4E B2RXH2 5/20 0.44
GAA P10253 2/20 0.42
HPGD P15428 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
NOTUM Q6P988 1/20 0.40
POLB P06746 1/20 0.40
NQO2 P16083 1/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9340393 0.91 HSD17B10 (0.45) HSD17B10TPMTALDH1A1KDM4EGAA
SCHEMBL6775493 0.89 HSD17B10 (0.46) HSD17B10TPMTALDH1A1KDM4EGAA
SCHEMBL6772316 0.86 HSD17B10 (0.44) HSD17B10TPMTALDH1A1KDM4EGAA
SCHEMBL7321975 0.86 TPMT (0.46) HSD17B10TPMTALDH1A1KDM4EGAA
SCHEMBL11468821 0.86 HSD17B10 (0.47) HSD17B10TPMTALDH1A1KDM4EGAA
SCHEMBL7357713 0.85 HSD17B10 (0.42) HSD17B10TPMTALDH1A1KDM4EGAA
SCHEMBL7360614 0.85 HSD17B10 (0.42) HSD17B10TPMTALDH1A1KDM4EGAA
SCHEMBL8804900 0.84 TPMT (0.47) HSD17B10TPMTALDH1A1KDM4EGAA
SCHEMBL13255342 0.84 GAA (0.57) HSD17B10ALDH1A1KDM4EGAAHPGD
SCHEMBL5925643 0.82 ACHE (0.43) HSD17B10TPMTALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1990006309-A1 HETEROAZABENZOBICYCLIC CARBOXAMIDE 5-HT3, ANTAGONISTS RORER INTERNATIONAL (OVERSEAS) INC. (US) 1990-06-14 WO disclosed
US-4933445-A Heteroazabenzobicyclic carboxamide 5-HT3 antagonists RORER PHARMACEUTICAL CORPORATION (US) 1990-06-12 US disclosed