SCHEMBL7316533

SCHEMBL7316533

CCCc1[nH]cnc1CCC(=O)N(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
GABRR1 P24046 1/20 0.36
HRH2 P25021 1/20 0.34
HRH1 P35367 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
EGFR P00533 1/20 0.33
SRC P12931 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HTR3E A5X5Y0 2/20 0.33
HTR3B O95264 2/20 0.33
HTR3A P46098 2/20 0.33
HTR3D Q70Z44 2/20 0.33
HTR3C Q8WXA8 2/20 0.33
NR4A1 P22736 1/20 0.33
NR4A2 P43354 1/20 0.33
NR4A3 Q92570 1/20 0.33
HSD17B10 Q99714 2/20 0.33
CYP2C19 P33261 2/20 0.33
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7266119 0.81 HRH4 (0.56) GABRR1HRH2HRH1HRH4HRH3
Hydrochloric Acid SCHEMBL7274987 0.79 TDP1 (0.57) GABRR1HRH2HRH1HRH4HRH3
SCHEMBL28285468 0.77 HRH3 (0.42) GABRR1HRH2HRH1HRH4HRH3
SCHEMBL7312965 0.72 HRH3 (0.38) GABRR1HRH2HRH1HRH4HRH3
SCHEMBL23418438 0.72 HRH3 (0.41) GABRR1HRH2HRH1HRH4HRH3
Hydrochloric Acid SCHEMBL7313845 0.71 TDP1 (0.40) GABRR1HRH2HRH1HRH4HRH3
SCHEMBL14290737 0.70 HRH3 (0.39) GABRR1HRH2HRH1HRH4HRH3
SCHEMBL10728091 0.69 HRH3 (0.47) HRH2HRH1HRH4HRH3TDP1
SCHEMBL721194 0.67 HRH3 (0.41) HRH2HRH1HRH4HRH3TDP1
SCHEMBL7316202 0.67 MAP3K7 (0.36) ALDH1A1NR4A2HSD17B10CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0242973-B1 INDOLE DERIVATIVES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1991-07-17 EP disclosed
US-4808581-A ANXIOLYTIC, ANTIEMETIC, TREATMENT OF PSYCHOLOGICAL DISORDERS GLAXO GROUP LIMITED (GB) 1989-02-28 US disclosed
EP-0242973-A1 Indole derivatives, method for their preparation and pharmaceutical compositions containing them GLAXO GROUP LIMITED (GB) 1987-10-28 EP disclosed