SCHEMBL7316202

SCHEMBL7316202

CCCc1[nH]cnc1C=CC(=O)N(C)C

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP3K7 O43318 1/20 0.36
TAB1 Q15750 1/20 0.36
SELP P16109 1/20 0.33
NR4A2 P43354 1/20 0.32
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
APP P05067 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7316193 1.00 MAP3K7 (0.36) MAP3K7TAB1SELPNR4A2CYP2C19
SCHEMBL7316533 0.67 ALDH1A1 (0.39) NR4A2CYP2C19HSD17B10NPC1ALDH1A1
SCHEMBL3953444 0.65 NR4A2 (0.38) MAP3K7TAB1NR4A2APP
SCHEMBL5870589 0.64 CYP2C19 (0.65) CYP2C19HSD17B10NPC1ALDH1A1MAPT
SCHEMBL7322217 0.64 MAP3K7 (0.37) MAP3K7TAB1NR4A2APP
SCHEMBL3003194 0.64 MAP3K7 (0.37) MAP3K7TAB1NR4A2APP
SCHEMBL6499135 0.63 CYP2C19 (0.44) CYP2C19HSD17B10ALDH1A1
SCHEMBL5870372 0.63 CYP2C19 (0.44) CYP2C19HSD17B10ALDH1A1MAPTKMT2A
Hydrochloric Acid SCHEMBL5869997 0.63 CYP2C19 (0.62) CYP2C19HSD17B10NPC1ALDH1A1MAPT
SCHEMBL24149480 0.62 NR4A2 (0.41) MAP3K7TAB1NR4A2APPNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0242973-B1 INDOLE DERIVATIVES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1991-07-17 EP disclosed
US-4808581-A ANXIOLYTIC, ANTIEMETIC, TREATMENT OF PSYCHOLOGICAL DISORDERS GLAXO GROUP LIMITED (GB) 1989-02-28 US disclosed
EP-0242973-A1 Indole derivatives, method for their preparation and pharmaceutical compositions containing them GLAXO GROUP LIMITED (GB) 1987-10-28 EP disclosed