SCHEMBL7318262

SCHEMBL7318262

CCCn1c(=O)c2[nH]c(-c3ccc(C(=N)N)cc3)nc2n(CCC)c1=O

nearest known ligand 0.81

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 14/20 0.81
ADORA2A P29274 7/20 0.81
ADORA1 P30542 1/20 0.73
KDM4E B2RXH2 2/20 0.69
MEN1 O00255 2/20 0.69
ALDH1A1 P00352 2/20 0.69
KMT2A Q03164 2/20 0.69
HSD17B10 Q99714 2/20 0.69
CYP1A2 P05177 1/20 0.69
CYP3A4 P08684 1/20 0.69
CYP2C9 P11712 1/20 0.69
CYP2C19 P33261 1/20 0.69
ADORA3 P0DMS8 3/20 0.67
GLA P06280 1/20 0.67
HPGD P15428 1/20 0.67
TSHR P16473 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7326027 0.99 ADORA2B (0.80) ADORA2BADORA2AADORA1KDM4EMEN1
Hydrochloric Acid SCHEMBL7315639 0.98 ADORA2B (0.78) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL7313469 0.87 ADORA2B (0.72) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL7313439 0.87 ADORA2B (0.72) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL7325450 0.86 ADORA2B (0.77) ADORA2BADORA2AADORA1KDM4EMEN1
Hydrochloric Acid SCHEMBL7316341 0.85 ADORA2B (0.70) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL7318202 0.84 ADORA2B (1.00) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL1948455 0.84 ADORA2B (1.00) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL7317209 0.84 ADORA2B (0.67) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL14564546 0.83 ADORA2B (0.79) ADORA2BADORA2AADORA1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0267607-B1 8-ARYLXANTHINES MARION MERRELL DOW INC. (US) 1991-11-27 EP disclosed
US-4783530-A CARDIOTONIC AND BRONCHODILATOR AGENTS MARION LABORATORIES, INC. (US) 1988-11-08 US disclosed
EP-0267607-A1 8-Arylxanthines MARION MERRELL DOW INC. (US) 1988-05-18 EP disclosed