SCHEMBL7319632

SCHEMBL7319632

O=C(O)C[C@@H](CCCc1ccccc1)C(=O)O

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.64
CPA1 P15085 2/20 0.62
CPB1 P15086 1/20 0.62
CPA3 P15088 1/20 0.62
CPB2 Q96IY4 1/20 0.62
MMP2 P08253 12/20 0.57
MMP3 P08254 4/20 0.57
HDAC3 O15379 1/20 0.53
MAPK1 P28482 1/20 0.53
ADRA1A P35348 1/20 0.53
HDAC4 P56524 1/20 0.53
SLC6A3 Q01959 1/20 0.53
HDAC1 Q13547 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC2 Q92769 1/20 0.53
HDAC10 Q969S8 1/20 0.53
HDAC11 Q96DB2 1/20 0.53
HDAC8 Q9BY41 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17537908 0.93 GRIK1 (0.54) GRIK1CPA1CPB1CPA3CPB2
SCHEMBL11311301 0.89 CPA1 (0.67) GRIK1CPA1CPB1CPA3CPB2
SCHEMBL9196227 0.89 CPA1 (0.67) GRIK1CPA1CPB1CPA3CPB2
SCHEMBL10734883 0.89 CPA1 (0.67) GRIK1CPA1CPB1CPA3CPB2
SCHEMBL1856639 0.89 GRIK1 (0.72) GRIK1CPA1CPA3CPB2MMP2
SCHEMBL1860416 0.85 GRIK1 (0.68) GRIK1CPA3CPB2MMP2MMP3
SCHEMBL7366093 0.85 GRIK1 (0.59) GRIK1CPA1CPB1CPA3CPB2
SCHEMBL7861733 0.85 TSHR (0.66) GRIK1MMP2MMP3
SCHEMBL17693397 0.85 CA2 (0.50) GRIK1CPA1CPB1CPA3CPB2
SCHEMBL17537904 0.85 FOLH1 (0.61) GRIK1CPA1CPB1CPA3CPB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0561758-A2 Method of preparing optically active homo-beta-amino acids MONSANTO COMPANY (US) 1993-09-22 EP disclosed
US-5229420-A Renin inhibitor G. D. SEARLE & CO. (US) 1993-07-20 US disclosed
EP-0349921-A2 Etheral n-terminal aminodiol amino acid derivatives as anti-hypertensive agents G.D. Searle & Co. (US) 1990-01-10 EP disclosed