SCHEMBL7320224

SCHEMBL7320224

COc1ccc2c(c1)O[C@@H](C(=O)O)CC2

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.51
PPARA Q07869 4/20 0.51
PPARD Q03181 3/20 0.51
FFAR1 O14842 1/20 0.50
CYP4F2 P78329 5/20 0.47
CYP4A11 Q02928 5/20 0.47
CA2 P00918 2/20 0.47
CA5A P35218 1/20 0.47
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
POLA1 P09884 2/20 0.45
MTNR1A P48039 2/20 0.45
MTNR1B P49286 1/20 0.45
LTB4R Q15722 1/20 0.45
LTB4R2 Q9NPC1 1/20 0.45
CA1 P00915 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7320221 1.00 PPARG (0.51) PPARGPPARAPPARDFFAR1CYP4F2
SCHEMBL7320228 1.00 PPARG (0.51) PPARGPPARAPPARDFFAR1CYP4F2
SCHEMBL7296319 0.89 PPARG (0.51) PPARGPPARACYP4F2CYP4A11NFKB1
SCHEMBL7296313 0.89 PPARG (0.51) PPARGPPARACYP4F2CYP4A11NFKB1
SCHEMBL29586849 0.85 CYP4F2 (0.53) PPARGPPARAPPARDFFAR1CYP4F2
SCHEMBL7286847 0.85 GLS (0.46) PPARDFFAR1CA2CA5AMTNR1A
SCHEMBL7286852 0.85 GLS (0.46) PPARDFFAR1CA2CA5AMTNR1A
SCHEMBL431776 0.85 PPARG (0.58) PPARGPPARAPPARDFFAR1CYP4F2
SCHEMBL2133112 0.83 PPARG (0.65) PPARGPPARAPPARDCYP4F2CYP4A11
SCHEMBL7313848 0.83 CYP4F2 (0.60) PPARGPPARAPPARDFFAR1CYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684039-A Chroman-2-ylmethylamino derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1997-11-04 US disclosed
US-5670667-A DOPAMINE INHIBITORS FOR PSYCHOLOGICAL DISORDERS AMERICAN HOME PRODUCTS CORPORATION (US) 1997-09-23 US disclosed
US-5541199-A DOPAMINE MODULATORS, SCHIZOPHRENIA AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-30 US disclosed