SCHEMBL7322182

SCHEMBL7322182

O=C(O)c1ccc(-c2nnc(-c3ccc(OCCCCOc4ccccc4)cc3)s2)cc1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.66
HDAC1 Q13547 6/20 0.65
HDAC2 Q92769 6/20 0.65
HDAC6 Q9UBN7 4/20 0.64
PKM P14618 1/20 0.62
RARB P10826 4/20 0.56
HDAC8 Q9BY41 3/20 0.55
PLA2G4B P0C869 1/20 0.53
CSNK2A2 P19784 3/20 0.53
CSNK2A1 P68400 3/20 0.53
TP53 P04637 1/20 0.52
TSHR P16473 1/20 0.52
CSNK2B P67870 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7321811 0.99 HDAC1 (0.66) NR1H4HDAC1HDAC2HDAC6PKM
SCHEMBL6538522 0.97 NR1H4 (0.66) NR1H4HDAC1HDAC2HDAC6PKM
SCHEMBL5969241 0.89 RARB (0.72) NR1H4RARBPLA2G4BCSNK2A2CSNK2A1
SCHEMBL6539365 0.89 NR1H4 (0.70) NR1H4RARBPLA2G4BCSNK2A2CSNK2A1
SCHEMBL7316607 0.88 NR1H4 (0.65) NR1H4HDAC1HDAC2HDAC6RARB
SCHEMBL7341006 0.88 NR1H4 (0.65) NR1H4HDAC1HDAC2HDAC6RARB
SCHEMBL7332564 0.88 RARB (0.75) NR1H4RARBPLA2G4BCSNK2A2CSNK2A1
SCHEMBL7317106 0.88 NR1H4 (0.65) NR1H4HDAC1HDAC2HDAC6RARB
SCHEMBL6539567 0.88 RARB (0.75) NR1H4RARBPLA2G4BCSNK2A2CSNK2A1
SCHEMBL7316179 0.88 NR1H4 (0.65) NR1H4HDAC1HDAC2HDAC6RARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6232290-B1 FUNGICIDES AGAINST PNEUMOCYSTIS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-15 US disclosed
EP-1053247-A1 ANTIFUNGAL CYCLOHEXAPEPTIDES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-11-22 EP disclosed
WO-1999040108-A1 NEW COMPOUND FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-08-12 WO disclosed