SCHEMBL7322337

SCHEMBL7322337

CON(C(=O)c1ccc(C(=O)NO)cc1)c1ccc2occc2c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
HTR1B P28222 1/20 0.41
CTNNB1 P35222 4/20 0.41
WNT3A P56704 4/20 0.41
HDAC6 Q9UBN7 8/20 0.39
HDAC1 Q13547 3/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
HDAC8 Q9BY41 4/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
IDO1 P14902 2/20 0.38
NAMPT P43490 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7321077 0.80 HDAC1 (0.47) HDAC6HDAC1CA1CA2HDAC8
SCHEMBL7311746 0.76 HDAC8 (0.53) CTNNB1WNT3AHDAC6HDAC1CA1
SCHEMBL14880251 0.76 HTR1B (0.56) TAS1R3TAS1R1HTR1BCTNNB1WNT3A
SCHEMBL7309720 0.75 HDAC6 (0.43) HDAC6HDAC1CA1CA2HDAC3
SCHEMBL7322358 0.74 HDAC6 (0.46) HDAC6HDAC1HDAC8HDAC3HDAC2
SCHEMBL7319461 0.74 CA1 (0.38) HDAC6HDAC1CA1CA2HDAC8
SCHEMBL7314295 0.73 HDAC6 (0.46) HDAC6HDAC1CA1CA2HDAC8
SCHEMBL7320946 0.72 HDAC6 (0.58) HDAC6HDAC1HDAC8HDAC3HDAC2
SCHEMBL1922481 0.70 CTNNB1 (0.50) TAS1R3TAS1R1HTR1BCTNNB1WNT3A
SCHEMBL30446573 0.70 CTNNB1 (0.50) TAS1R3TAS1R1HTR1BCTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230094176-A1 COMPOUNDS AND METHODS FOR IMPROVING IMPAIRED ENDOGENOUS FIBRINOLYSIS USING HISTONE DEACETYLASE INHIBITORS CERENO SCIENT AB (SE) 2023-03-30 US disclosed
US-20210060014-A1 COMPOUNDS AND METHODS FOR IMPROVING IMPAIRED ENDOGENOUS FIBRINOLYSIS USING HISTONE DEACETYLASE INHIBITORS CERENO SCIENTIFIC AB (SE) 2021-03-04 US disclosed
US-20170020874-A1 COMPOUNDS AND METHODS FOR IMPROVING IMPAIRED ENDOGENOUS FIBRINOLYSIS USING HISTONE DEACETYLASE INHIBITORS CERENO SCIENT AB (SE) 2017-01-26 US disclosed
EP-0901465-B1 COMPOUNDS WITH ANTI-INFLAMMATORY AND IMMUNOSUPPRESSIVE ACTIVITIES ITALFARMACO SPA (IT) 2000-09-27 EP disclosed
US-6034096-A Compounds with anti-inflammatory and immunosuppressive activities ITALFARMACO S.P.A. (IT) 2000-03-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170020874-A1 COMPOUNDS AND METHODS FOR IMPROVING IMPAIRED ENDOGENOUS FIBRINOLYSIS USING HISTONE DEACETYLASE INHIBITORS HDAC3, HDAC1, HDAC2 TAS1R3 4242/4885TAS1R1 4465/4885HTR1B 4259/4885
US-20210060014-A1 COMPOUNDS AND METHODS FOR IMPROVING IMPAIRED ENDOGENOUS FIBRINOLYSIS USING HISTONE DEACETYLASE INHIBITORS HDAC3, HDAC1, HDAC2 TAS1R3 4242/4885TAS1R1 4465/4885HTR1B 4259/4885
US-20230094176-A1 COMPOUNDS AND METHODS FOR IMPROVING IMPAIRED ENDOGENOUS FIBRINOLYSIS USING HISTONE DEACETYLASE INHIBITORS HDAC3, HDAC2, HDAC1 TAS1R3 4335/4885TAS1R1 4592/4885HTR1B 4013/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.