SCHEMBL7322773

SCHEMBL7322773

Cc1coc(C)c1-c1nc2cc(Cl)cc(CCc3ccccn3)c2o1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KDM4E B2RXH2 7/20 0.34
ALDH1A1 P00352 6/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
HSD17B10 Q99714 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
CETP P11597 2/20 0.34
MAPT P10636 2/20 0.34
RECQL P46063 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
ATM Q13315 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7325321 0.80 ADORA2A (0.49) CYP2D6CYP1A2TDP1KDM4EALDH1A1
SCHEMBL7322971 0.80 NPC1 (0.41) CYP2D6CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL7314123 0.79 KDM4E (0.37) CYP2D6CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL7325292 0.79 KDM4E (0.34) CYP2D6CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL7316469 0.78 KDM4E (0.35) CYP2D6CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL7323231 0.78 ALDH1A1 (0.43) CYP2C19CYP1A2KDM4EALDH1A1NPC1
SCHEMBL7315804 0.78 ALDH1A1 (0.36) CYP2D6CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL7322017 0.78 HSP90AA1 (0.36) CYP2D6CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL7317091 0.77 PDGFRB (0.38) KDM4EALDH1A1NPC1RAB9AHSD17B10
SCHEMBL7324311 0.77 KDM4E (0.40) CYP2D6CYP2C9CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166041-A 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma EURO-CELTIQUE, S.A. (LU) 2000-12-26 US claimed
US-6166041-A 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma EURO-CELTIQUE, S.A. (LU) 2000-12-26 US disclosed