SCHEMBL7324466

SCHEMBL7324466

OC1(Cl)C=CC(C=Cc2ccccc2)=CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.37
TTR P02766 1/20 0.35
ALOX5 P09917 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
CHAT P28329 1/20 0.33
MEN1 O00255 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAOB P27338 2/20 0.32
NFE2L2 Q16236 1/20 0.32
CYP19A1 P11511 1/20 0.32
MAOA P21397 1/20 0.32
PTPN1 P18031 1/20 0.32
HNF4A P41235 1/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC3 O15379 1/20 0.32
TNKS O95271 1/20 0.32
HDAC4 P56524 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2532692 0.83 TTR (0.37) TRPA1TTRALOX5PTGS1PTGS2
SCHEMBL28697334 0.83 CHAT (0.35) TRPA1TTRALOX5PTGS1PTGS2
SCHEMBL27693757 0.82 MAOB (0.37) TRPA1TTRALOX5PTGS1PTGS2
SCHEMBL9344854 0.82 MAOB (0.37) TRPA1TTRALOX5PTGS1PTGS2
SCHEMBL29036461 0.79 LCK (0.44) TRPA1TTRALOX5PTGS1PTGS2
SCHEMBL27570573 0.78 HDAC1 (0.37) TTRALOX5PTGS1PTGS2MEN1
SCHEMBL4438933 0.78 MAOB (0.39) TRPA1TTRALOX5PTGS1PTGS2
SCHEMBL27790759 0.78 MAPT (0.45) MEN1MAPTKMT2AMAOBCYP19A1
SCHEMBL9546943 0.77 HDAC1 (0.36) TTRALOX5PTGS1PTGS2MAPT
SCHEMBL2905608 0.77 TTR (0.36) TRPA1TTRALOX5PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625979-A1 AZABRICYCLIC COMPOUNDS AS CALCIUM CHANNEL ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-11-30 EP disclosed
WO-1993015073-A1 AZABRICYCLIC COMPOUNDS AS CALCIUM CHANNEL ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-08-05 WO disclosed