SCHEMBL7324697

SCHEMBL7324697

CC(OC(=O)C(=O)CCc1ccccc1)N(C)C

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.46
KEAP1 Q14145 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PLAAT5 Q96KN8 3/20 0.43
PLAAT4 Q9UL19 3/20 0.43
FFAR1 O14842 2/20 0.42
ALOX5 P09917 1/20 0.42
TSHR P16473 1/20 0.41
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
PLAAT3 P53816 2/20 0.41
PLAAT2 Q9NWW9 2/20 0.41
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058635 0.84 TSHR (0.54) KMT2AMEN1ALDH1A1KEAP1TDP1
SCHEMBL7061795 0.80 ALDH1A1 (0.47) KMT2AMEN1ALDH1A1KEAP1TDP1
SCHEMBL991969 0.75 ALDH1A1 (0.57) ALDH1A1KEAP1TDP1PLAAT5PLAAT4
SCHEMBL7641654 0.75 HDAC1 (0.53) KMT2ATDP1PLAAT5PLAAT4TSHR
SCHEMBL7061750 0.75 TDP1 (0.50) KMT2AMEN1ALDH1A1KEAP1TDP1
Hydrochloric Acid SCHEMBL5708139 0.75 TSHR (0.47) KMT2AALDH1A1ALOX5TSHRCHRNB2
SCHEMBL7641646 0.74 MAPT (0.53) KMT2AALDH1A1PLAAT5PLAAT4ALOX5
SCHEMBL10751276 0.73 TSHR (0.67) KMT2AALDH1A1TSHRCHRNB2CHRNB4
SCHEMBL7635416 0.73 MAPT (0.56) PLAAT5PLAAT4ALOX5TSHRPLAAT3
SCHEMBL7277555 0.73 CHRM1 (0.52) KMT2AALDH1A1KEAP1TDP1PLAAT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4472380-A CARBOXYALKYL DIPEPTIDE DERIVATIVES MERCK & CO., INC. (US) 1984-09-18 US disclosed
US-4374829-A Aminoacid derivatives as antihypertensives MERCK & CO., INC. (US) 1983-02-22 US disclosed
EP-0012401-A1 Carboxyalkyl dipeptide derivatives, process for preparing them and pharmaceutical composition containing them MERCK & CO. INC. (US) 1980-06-25 EP disclosed