Dexamethasone

Dexamethasone

SCHEMBL73250

C[C@@H]1C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO.O=P(O)(O)O

nearest known ligand 0.93

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Dexamethasone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 7/20 0.93
HIF1A Q16665 9/20 0.93
CYP3A4 P08684 7/20 0.93
HSD17B10 Q99714 4/20 0.93
NFKB1 P19838 3/20 0.93
PGR P06401 3/20 0.93
TSHR P16473 2/20 0.93
AR P10275 2/20 0.93
PMP22 Q01453 2/20 0.93
MEN1 O00255 1/20 0.93
CYP2D6 P10635 1/20 0.93
KMT2A Q03164 1/20 0.93
APEX1 P27695 1/20 0.93
NPSR1 Q6W5P4 1/20 0.93
IKBKB O14920 1/20 0.93
CHUK O15111 1/20 0.93
ADRB2 P07550 1/20 0.93
NR3C2 P08235 1/20 0.93
PLA2G2A P14555 1/20 0.93
NFKB2 Q00653 1/20 0.93

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Betamethasone SCHEMBL7426 1.00 HIF1A (0.93) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Dexamethasone SCHEMBL4973562 1.00 HIF1A (0.93) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Dexamethasone SCHEMBL1561578 1.00 HIF1A (0.93) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Betamethasone SCHEMBL5501682 1.00 HIF1A (0.93) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Betamethasone SCHEMBL27476350 1.00 HIF1A (0.93) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Betamethasone SCHEMBL8529637 1.00 HIF1A (0.93) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Betamethasone SCHEMBL28777880 0.99 HIF1A (0.92) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Betamethasone SCHEMBL1479323 0.99 HIF1A (0.92) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Betamethasone SCHEMBL2807697 0.99 HIF1A (0.92) HIF1ACYP3A4NR3C1HSD17B10NFKB1
Dexamethasone SCHEMBL2808007 0.99 HIF1A (0.92) HIF1ACYP3A4NR3C1HSD17B10NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4296 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121490062-B Dexamethasone-containing composition and application thereof in preparation of medicament for treating retinopathy 上饶爱尔眼科医院有限公司 2026-05-15 CN claimed
US-20260108657-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATING OSTEOARTHRITIS INSIGNIA PHARMACEUTICALS, LLC (US) 2026-04-23 US claimed
US-12551148-B2 Systems and methods for compensating for agent elution MEDTRONIC MINIMED, INC. (US) 2026-02-17 US claimed
US-20260021113-A1 INTRAVITREAL CORTICOSTEROID EXTENDED RELEASE IMPLANT AND METHODS OF USE EYEDEA BIO LLC (US) 2026-01-22 US claimed
US-12491289-B2 Pharmaceutical compositions for treating osteoarthritis INSIGNIA PHARMACEUTICALS, LLC (US) 2025-12-09 US claimed
EP-4654956-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATING OSTEOARTHRITIS Insignia Pharmaceuticals, LLC (US) 2025-12-03 EP claimed
US-12433900-B2 Intravitreal corticosteroid extended release implant and methods of use EYEDEA BIO, LLC (US) 2025-10-07 US claimed
US-20250295608-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR TREATING OSTEOARTHRITIS INSIGNIA PHARMACEUTICALS, LLC (US) 2025-09-25 US claimed
US-20250288599-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR TREATING OSTEOARTHRITIS INSIGNIA PHARMACEUTICALS, LLC (US) 2025-09-18 US claimed
US-20250275916-A1 MEDICATED EYELID CLEANSING COMPOSITIONS OCUSOFT, INC. 2025-09-04 US claimed
EP-0622090-A1 Sintered electrode on a substrate MEDTRONIC, INC. (US) 1994-11-02 EP claimed
US-5282844-A High impedance, low polarization, low threshold miniature steriod eluting pacing lead electrodes MEDTRONIC, INC. (US) 1994-02-01 US claimed
US-5232441-A Method of treating schistosomal infestations by iontophoresis PHYSION S.R.L. (IT) 1993-08-03 US claimed
CN-1073859-A Regulate the compositions of wrinkle of skin and/or atrophoderma RICHARDSON VICKS INC (US) 1993-07-07 CN claimed
EP-0538368-A1 MINIATURE STEROID ELUTING PACING LEAD ELECTRODE MEDTRONIC, INC. (US) 1993-04-28 EP claimed
WO-1991019533-A1 MINIATURE STEROID ELUTING PACING LEAD ELECTRODE MEDTRONIC, INC. (US) 1991-12-26 WO claimed
US-4506680-A Drug dispensing body implantable lead MEDTRONIC, INC. (US) 1985-03-26 US claimed
US-4346709-A Drug delivery devices comprising erodible polymer and erosion rate modifier ALZA CORPORATION (US) 1982-08-31 US claimed
EP-0056420-A1 Ophthalmic gel SCHERING CORPORATION (US) 1982-07-28 EP claimed
US-4255415-A COMPRISING A MEDICAMENT, A VINYL ACETATE-VINYL ALCOHOL COPOLYMER, AN ALKALI OR ALKALINE BORATE, AND STERILE WATER; TOPICAL SCHERING CORPORATION (US) 1981-03-10 US claimed