SCHEMBL7325199

SCHEMBL7325199

CCCn1c(=O)c2[nH]c(-c3ccc(C#N)cc3)nc2n(CCC)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 14/20 0.72
ADORA2A P29274 6/20 0.72
ADORA1 P30542 3/20 0.72
KDM4E B2RXH2 2/20 0.72
CYP1A2 P05177 2/20 0.72
CYP3A4 P08684 2/20 0.72
MEN1 O00255 1/20 0.72
ALDH1A1 P00352 1/20 0.72
CYP2C9 P11712 1/20 0.72
CYP2C19 P33261 1/20 0.72
KMT2A Q03164 1/20 0.72
HSD17B10 Q99714 1/20 0.72
ADORA3 P0DMS8 2/20 0.71
LMNA P02545 1/20 0.71
THRB P10828 1/20 0.71
BLM P54132 1/20 0.71
PMP22 Q01453 1/20 0.71
NPSR1 Q6W5P4 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323908 0.93 ADORA2B (0.64) ADORA2BADORA2AADORA1KDM4ECYP1A2
SCHEMBL7325375 0.93 ADORA2B (0.66) ADORA2BADORA2AADORA1KDM4ECYP1A2
SCHEMBL14564546 0.85 ADORA2B (0.79) ADORA2BADORA2AADORA1KDM4ECYP1A2
SCHEMBL14875118 0.85 ADORA2B (0.77) ADORA2BADORA2AADORA1KDM4ECYP1A2
Water SCHEMBL15690379 0.84 ADORA2B (1.00) ADORA2BADORA2AADORA1KDM4ECYP1A2
SCHEMBL1222380 0.84 ADORA2B (1.00) ADORA2BADORA2AADORA1KDM4ECYP1A2
SCHEMBL7318202 0.84 ADORA2B (1.00) ADORA2BADORA2AADORA1KDM4ECYP1A2
SCHEMBL1948455 0.84 ADORA2B (1.00) ADORA2BADORA2AADORA1KDM4ECYP1A2
SCHEMBL1943831 0.84 ADORA2B (0.79) ADORA2BADORA2AADORA1ADORA3
SCHEMBL661108 0.84 ADORA2B (1.00) ADORA2BADORA2AADORA1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0267607-B1 8-ARYLXANTHINES MARION MERRELL DOW INC. (US) 1991-11-27 EP disclosed
US-4783530-A CARDIOTONIC AND BRONCHODILATOR AGENTS MARION LABORATORIES, INC. (US) 1988-11-08 US disclosed
EP-0267607-A1 8-Arylxanthines MARION MERRELL DOW INC. (US) 1988-05-18 EP disclosed