SCHEMBL7325359

SCHEMBL7325359

Cn1c(=O)c2[nH]c(-c3ccc(C#N)cc3)nc2n(C)c1=O

nearest known ligand 0.74

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 5/20 0.70
ADORA2A P29274 3/20 0.70
KDM4E B2RXH2 2/20 0.69
ADORA1 P30542 2/20 0.69
CYP1A2 P05177 1/20 0.69
ADORA3 P0DMS8 1/20 0.69
BLM P54132 1/20 0.69
NPSR1 Q6W5P4 1/20 0.69
HSD17B10 Q99714 1/20 0.69
ALDH1A1 P00352 1/20 0.67
HPGD P15428 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL7315528 1.00 ADORA2B (0.70) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL7325375 0.86 ADORA2B (0.66) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL7323908 0.86 ADORA2B (0.64) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL25090525 0.85 ADORA2B (0.67) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL516013 0.83 ADORA2B (0.77) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL10723936 0.82 ADORA2B (1.00) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL515588 0.82 KDM4E (0.76) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL25090491 0.82 ADORA2B (0.75) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL516029 0.82 ADORA2B (0.75) ADORA2BADORA2AKDM4EADORA1CYP1A2
SCHEMBL7318169 0.82 KDM4E (0.76) ADORA2BADORA2AKDM4EADORA1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0267607-B1 8-ARYLXANTHINES MARION MERRELL DOW INC. (US) 1991-11-27 EP disclosed
US-4783530-A CARDIOTONIC AND BRONCHODILATOR AGENTS MARION LABORATORIES, INC. (US) 1988-11-08 US disclosed
EP-0267607-A1 8-Arylxanthines MARION MERRELL DOW INC. (US) 1988-05-18 EP disclosed