Oxalic Acid

Oxalic Acid

SCHEMBL7325487

C#CC1(OCc2ccccc2F)CCN(C)CC1.O=C(O)C(=O)O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 3/20 0.38
SLC6A4 known ✓ P31645 1/20 0.38
KMT2A Q03164 5/20 0.43
MEN1 O00255 3/20 0.43
RAB9A P51151 2/20 0.43
DPP4 P27487 1/20 0.42
ALDH1A1 P00352 6/20 0.40
KDM4E B2RXH2 3/20 0.40
MAPK1 P28482 2/20 0.40
ATM Q13315 2/20 0.38
SCN1A P35498 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
SLC22A1 O15245 1/20 0.38
ADRA1A P35348 1/20 0.38
KCNH2 Q12809 1/20 0.38
NPSR1 Q6W5P4 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10632013 0.93 CARM1 (0.38) KMT2AMEN1RAB9ADPP4ALDH1A1
SCHEMBL7330260 0.85 RAB9A (0.57) KMT2AMEN1RAB9ADPP4ALDH1A1
SCHEMBL11128101 0.84 RAB9A (0.56) KMT2AMEN1RAB9ADPP4ALDH1A1
SCHEMBL11128097 0.83 RAB9A (0.55) KMT2AMEN1RAB9ADPP4ALDH1A1
Oxalic Acid SCHEMBL7324471 0.82 KMT2A (0.48) KMT2AMEN1RAB9ADPP4ALDH1A1
SCHEMBL7334571 0.79 KMT2A (0.47) KMT2AMEN1RAB9ADPP4ALDH1A1
Oxalic Acid SCHEMBL7329943 0.79 DPP4 (0.44) KMT2AMEN1RAB9ADPP4ALDH1A1
SCHEMBL12050012 0.74 SCN1A (0.42) KMT2AMEN1RAB9ADPP4ALDH1A1
SCHEMBL7324921 0.74 RAB9A (0.41) KMT2AMEN1RAB9ADPP4ALDH1A1
SCHEMBL7323828 0.74 RAB9A (0.41) KMT2AMEN1RAB9ADPP4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0102034-B1 SPIRO(2H-1,4-BENZODIOXEPIN-3(5H)4'-PIPERIDINE AND 3'-PYRROLIDINO) COMPOUNDS, A PROCESS FOR PREPARING THE SAME AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1988-04-20 EP disclosed
US-4695637-A HYPOTENSIVE AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-09-22 US disclosed
US-4668791-A HYPOTENSIVE, ALDEHYDES HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-05-26 US disclosed
US-4579950-A HYPOTENSIVE AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-04-01 US disclosed
US-4577026-A HYPOTENSIVE AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-03-18 US disclosed
US-4569998-A HYPOTENSIVE AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-02-11 US disclosed
US-4521537-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1985-06-04 US disclosed
US-4472580-A Spiro (2H-1,4-benzodioxepin-3 (5H)4-piperidine and -3-pyrrolidine) compounds and their use as anti-hypertensive agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1984-09-18 US disclosed
US-4405631-A Spiro[2H-1,4-benzodioxepin-3(5H)4'-piperidine and -3'pyrrolidine] compounds and their use as antihypertensive agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1983-09-20 US disclosed