SCHEMBL7326240

SCHEMBL7326240

CCOC(=O)c1cn2cc(Br)nc(NC)c2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
POLB P06746 2/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
GAA P10253 1/20 0.40
CYP1A2 P05177 1/20 0.40
GABRA2 P47869 5/20 0.39
GABRB2 P47870 5/20 0.39
RXFP1 Q9HBX9 2/20 0.38
NPC1 O15118 2/20 0.38
MAPT P10636 2/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
EED O75530 1/20 0.37
RBBP4 Q09028 1/20 0.37
SUZ12 Q15022 1/20 0.37
EZH2 Q15910 1/20 0.37
AEBP2 Q6ZN18 1/20 0.37
CDC7 O00311 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31210678 0.84 KDM4E (0.49) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL7354451 0.84 KDM4E (0.49) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL23534393 0.81 KDM4E (0.46) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL7319485 0.80 SMN1; SMN2 (0.39) KDM4EPOLBALDH1A1GAACYP1A2
SCHEMBL13764178 0.80 KDM4E (0.54) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL29772651 0.79 KDM4E (0.36) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL25397343 0.76 MAPK1 (0.50) KDM4EPOLBALDH1A1HPGDCYP1A2
SCHEMBL31210467 0.76 KDM4E (0.49) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL5554280 0.76 KMT2A (0.49) KDM4EPOLBALDH1A1HPGDGAA
SCHEMBL29772664 0.76 MERTK (0.39) KDM4EPOLBALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5028605-A Antispasmodic, bronchodilators, uterine relaxants, cardiac analeptics, neurosedatives L'UNIVERSITE DE MONTPELLIER I (FR) 1991-07-02 US disclosed
EP-0348392-A1 8-ALKYLAMINOIMIDAZO[1,2-A]PYRAZINES AND DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY Université Montpellier I (FR) 1990-01-03 EP disclosed
WO-1988004298-A1 8-ALKYLAMINOIMIDAZO[1,2-A]PYRAZINES AND DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1988-06-16 WO disclosed