SCHEMBL7326253

SCHEMBL7326253

OC1=Nc2ccccc2C2=NCCN12

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 1/20 0.51
RAD52 P43351 1/20 0.51
UHRF1 Q96T88 1/20 0.51
HDAC8 Q9BY41 5/20 0.49
HDAC4 P56524 2/20 0.49
PTAFR P25105 11/20 0.47
SMARCA2 P51531 1/20 0.43
EED O75530 1/20 0.42
HDAC5 Q9UQL6 1/20 0.41
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL86872 0.81 DNMT1 (0.53) DNMT1RAD52UHRF1HDAC8HDAC4
SCHEMBL7326935 0.80 DNMT1 (0.51) DNMT1RAD52UHRF1HDAC8HDAC4
Bromide SCHEMBL82425 0.80 DNMT1 (0.51) DNMT1RAD52UHRF1HDAC8HDAC4
SCHEMBL86484 0.75 PIK3CB (0.44) DNMT1RAD52UHRF1HDAC8HDAC4
SCHEMBL86777 0.74 DNMT1 (0.40) DNMT1RAD52UHRF1HDAC8HDAC4
SCHEMBL86897 0.74 DNMT1 (0.42) DNMT1RAD52UHRF1HDAC8HDAC4
SCHEMBL86781 0.73 DNMT1 (0.41) DNMT1RAD52UHRF1HDAC8HDAC4
SCHEMBL86500 0.73 PTAFR (0.42) DNMT1RAD52UHRF1HDAC8HDAC4
SCHEMBL86871 0.73 PIK3CB (0.46) DNMT1RAD52UHRF1HDAC8HDAC4
SCHEMBL87166 0.73 DNMT1 (0.41) DNMT1RAD52UHRF1HDAC8HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0491814-B1 TETRACYCLIC IMIDAZOQUINAZOLINE DERIVATIVES, PREPARATION AND PHARMACEUTICAL COMPOSITIONS NOVO NORDISK AS (DK) 1995-12-06 EP disclosed
US-5100895-A Imidazoquinazoline compounds; anticonvulsants, anxiolytics, hypnotics, antipsychotics, antiemetics, improving cognitive function NOVO NORDISK A/S (DK) 1992-03-31 US disclosed
EP-0417027-A1 Tetracyclic imidazoquinazoline derivatives, process for their preparation and pharmaceutical compositions containing them NOVO NORDISK A/S (DK) 1991-03-13 EP disclosed