SCHEMBL7326643

SCHEMBL7326643

CN1C(=O)CN(CCC(=O)O)C(=O)c2cc(C#Cc3ccc(CN)cc3)ccc21

nearest known ligand 0.75

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.75
ITGA2B P08514 6/20 0.75
KDM4E B2RXH2 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
FFAR1 O14842 10/20 0.38
HDAC1 Q13547 3/20 0.37
HDAC6 Q9UBN7 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7325747 0.94 ITGB3 (0.68) ITGB3ITGA2BKDM4EALOX15TSHR
Trifluoroacetic Acid SCHEMBL8959450 0.87 ITGB3 (0.66) ITGB3ITGA2BFFAR1
SCHEMBL8837187 0.86 ITGB3 (1.00) ITGB3ITGA2BKDM4EALOX15TSHR
SCHEMBL7325755 0.84 ITGB3 (0.56) ITGB3ITGA2BFFAR1HDAC1HDAC6
SCHEMBL7359324 0.84 ITGB3 (0.84) ITGB3ITGA2BKDM4EALOX15TSHR
Trifluoroacetic Acid SCHEMBL7324537 0.82 ITGB3 (0.69) ITGB3ITGA2BFFAR1HDAC1
Trifluoroacetic Acid SCHEMBL7320877 0.81 ITGB3 (0.90) ITGB3ITGA2BKDM4EALOX15TSHR
Trifluoroacetic Acid SCHEMBL8959447 0.81 ITGB3 (0.66) ITGB3ITGA2BKDM4EALOX15TSHR
Trifluoroacetic Acid SCHEMBL7322477 0.80 ITGB3 (0.61) ITGB3ITGA2BKDM4EALOX15TSHR
Ethyl Acetate SCHEMBL7330809 0.79 ITGB3 (0.85) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993008174-A1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPIIbIIIa RECEPTOR GENENTECH, INC. (US) 1993-04-29 WO disclosed