SCHEMBL7327014

SCHEMBL7327014

COc1ccc(CCN(C)CCCN(C(=O)c2ccc(N)cc2)c2ccc(OC)c(OC)c2)cc1OC

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.76
CYP3A4 P08684 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
SMPD1 P17405 3/20 0.53
BLM P54132 1/20 0.52
PMP22 Q01453 1/20 0.52
CYP19A1 P11511 1/20 0.47
ALDH1A1 P00352 3/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
ABCB1 P08183 1/20 0.46
AOC3 Q16853 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MAPT P10636 3/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9113987 0.99 KCNH2 (0.75) KCNH2CYP3A4CYP1A2CYP2D6SMPD1
SCHEMBL7265181 0.90 KCNH2 (0.76) KCNH2CYP3A4CYP1A2CYP2D6SMPD1
SCHEMBL7328234 0.90 KCNH2 (0.75) KCNH2CYP3A4CYP1A2CYP2D6SMPD1
SCHEMBL7333091 0.88 KCNH2 (0.73) KCNH2CYP3A4CYP1A2CYP2D6SMPD1
SCHEMBL7359612 0.87 KCNH2 (0.72) KCNH2CYP3A4CYP1A2CYP2D6SMPD1
SCHEMBL30357973 0.86 KCNH2 (1.00) KCNH2CYP3A4CYP1A2CYP2D6SMPD1
SCHEMBL9114669 0.86 KCNH2 (0.71) KCNH2CYP3A4CYP1A2CYP2D6SMPD1
Hydrochloric Acid SCHEMBL7333187 0.85 KCNH2 (0.98) KCNH2CYP3A4CYP1A2CYP2D6SMPD1
SCHEMBL7327022 0.85 KCNH2 (0.56) KCNH2CYP19A1ALDH1A1KMT2AMEN1
SCHEMBL9113035 0.85 KCNH2 (0.69) KCNH2CYP3A4CYP1A2CYP2D6SMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639973-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1995-03-01 EP claimed
WO-1993023024-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1993-11-25 WO claimed
EP-0852142-A1 Diamines in the treatment of arrhythmia SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1998-07-08 EP disclosed
EP-0639973-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1995-03-01 EP disclosed
WO-1993023024-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1993-11-25 WO disclosed