SCHEMBL7333091

SCHEMBL7333091

COc1ccc(CCN(C)CCCN(C(=O)c2ccncc2)c2ccc(OC)c(OC)c2)cc1OC

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.73
KDM4E B2RXH2 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
CYP3A4 P08684 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
SMPD1 P17405 3/20 0.53
BLM P54132 1/20 0.52
PMP22 Q01453 1/20 0.52
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 2/20 0.46
MAPT P10636 2/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
ABCB1 P08183 1/20 0.43
HCN4 Q9Y3Q4 1/20 0.43
SCN1A P35498 1/20 0.43
SCN2A Q99250 1/20 0.43
SCN3A Q9NY46 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7328234 0.90 KCNH2 (0.75) KCNH2KDM4ECYP3A4CYP1A2CYP2D6
SCHEMBL7265181 0.88 KCNH2 (0.76) KCNH2KDM4ECYP3A4CYP1A2CYP2D6
SCHEMBL7327014 0.88 KCNH2 (0.76) KCNH2KDM4ESMN1; SMN2CYP3A4CYP1A2
Hydrochloric Acid SCHEMBL9113987 0.87 KCNH2 (0.75) KCNH2KDM4ESMN1; SMN2CYP3A4CYP1A2
SCHEMBL9238469 0.86 KCNH2 (0.65) KCNH2KDM4ESMN1; SMN2CYP3A4CYP1A2
SCHEMBL7359612 0.85 KCNH2 (0.72) KCNH2SMN1; SMN2CYP3A4CYP1A2CYP2D6
SCHEMBL7333098 0.85 KCNH2 (0.54) KCNH2KDM4ESMN1; SMN2KMT2AALDH1A1
Hydrochloric Acid SCHEMBL678425 0.85 KCNH2 (0.96) KCNH2SMN1; SMN2CYP3A4CYP1A2CYP2D6
SCHEMBL9114669 0.84 KCNH2 (0.71) KCNH2SMN1; SMN2CYP3A4CYP1A2CYP2D6
SCHEMBL30357973 0.84 KCNH2 (1.00) KCNH2SMN1; SMN2CYP3A4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0852142-A1 Diamines in the treatment of arrhythmia SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1998-07-08 EP disclosed
EP-0639973-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1995-03-01 EP disclosed
WO-1993023024-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1993-11-25 WO disclosed