SCHEMBL7328197

SCHEMBL7328197

O=C(c1ccc(F)cc1)C1CCN(CCCl)CC1

nearest known ligand 0.72

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.72
HTR2C P28335 3/20 0.72
HTR7 P34969 3/20 0.72
HTR6 P50406 3/20 0.72
KDM4E B2RXH2 1/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2D6 P10635 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8403779 0.99 HTR2A (0.71) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL9726195 0.92 HTR2A (0.69) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL14318600 0.91 HTR2A (0.81) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL11516583 0.90 HTR2A (0.70) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL8714691 0.87 HTR2A (0.74) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL11747892 0.87 KCNH2 (0.64) HTR2AHTR2CHTR7HTR6
SCHEMBL10928970 0.85 HTR2A (0.72) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL9229261 0.85 HTR2A (0.72) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL10928975 0.85 HTR2A (0.72) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL20577435 0.85 HTR2A (0.71) HTR2AKDM4ECYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0841330-B1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-27 EP disclosed
US-5919784-A ANXIETY, DEPRESSION ADIR ET COMPAGNIE (FR) 1999-07-06 US disclosed
EP-0841330-A1 Aminomethyl heterocyclic derivatives, process of their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-05-13 EP disclosed
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed
US-5077288-A Adrenergic, serotonin and histamine antagonist ADIR ET COMPAGNIE (FR) 1991-12-31 US disclosed
US-4151285-A ANTICONVULSANT, ANTI-ANXIETY AGENTS A. H. ROBINS COMPANY, INC. (US) 1979-04-24 US disclosed
US-4032642-A SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1977-06-28 US disclosed
US-3956296-A ANTIINFLAMMATORY, SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1976-05-11 US disclosed