SCHEMBL7329638

SCHEMBL7329638

CC1CCc2cccc3c(C(=O)O)cn1c23

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
CYP1A2 P05177 1/20 0.57
CNR1 P21554 5/20 0.45
LMNA P02545 1/20 0.41
MCL1 Q07820 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CNR2 P34972 4/20 0.37
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
PDK1 Q15118 3/20 0.36
PDK2 Q15119 3/20 0.36
PDK3 Q15120 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3966675 0.91 KDM4E (0.67) KDM4ESMN1; SMN2CYP1A2CNR1LMNA
SCHEMBL3965154 0.91 KDM4E (0.67) KDM4ESMN1; SMN2CYP1A2CNR1LMNA
SCHEMBL6334232 0.83 KDM4E (0.44) KDM4ESMN1; SMN2CYP1A2CNR1LMNA
SCHEMBL3520185 0.80 CNR1 (0.64) KDM4ECNR1ALDH1A1GAAHPGD
SCHEMBL4129090 0.77 KDM4E (0.48) KDM4ESMN1; SMN2CYP1A2CNR1LMNA
SCHEMBL4129093 0.77 KDM4E (0.48) KDM4ESMN1; SMN2CYP1A2CNR1LMNA
SCHEMBL11257190 0.77 KDM4E (0.53) KDM4ESMN1; SMN2CYP1A2CNR1LMNA
SCHEMBL11741159 0.75 KDM4E (0.48) KDM4ESMN1; SMN2CYP1A2CNR1LMNA
SCHEMBL11745247 0.74 KDM4E (0.56) KDM4ESMN1; SMN2CYP1A2CNR1LMNA
SCHEMBL11750696 0.74 KDM4E (0.76) KDM4ESMN1; SMN2CYP1A2LMNAPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5102901-A 5-hydroxytrypamine receptor antaonists DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1992-04-07 US disclosed
EP-0393766-A2 New 3-N substituted carbamoyl-indole derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-10-24 EP disclosed