SCHEMBL7330385

SCHEMBL7330385

COc1ccc(OC)c(C(=O)/C=C/c2cccc(C(=O)O)c2)c1

nearest known ligand 0.77

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.70
PDE4A P27815 1/20 0.69
PDE4B Q07343 1/20 0.69
PDE4C Q08493 1/20 0.69
PDE4D Q08499 1/20 0.69
MEN1 O00255 1/20 0.62
NPC1 O15118 1/20 0.62
MAPT P10636 1/20 0.62
RAB9A P51151 1/20 0.62
KMT2A Q03164 1/20 0.62
BCHE P06276 1/20 0.61
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
MAOB P27338 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7330391 1.00 ABCG2 (0.70) ABCG2PDE4APDE4BPDE4CPDE4D
SCHEMBL28906337 0.88 NR1H4 (0.70) ABCG2MEN1NPC1MAPTRAB9A
SCHEMBL9982860 0.87 ABCG2 (0.86) ABCG2PDE4APDE4BPDE4CPDE4D
SCHEMBL9982858 0.87 ABCG2 (0.86) ABCG2PDE4APDE4BPDE4CPDE4D
SCHEMBL9986620 0.86 ABCG2 (0.84) ABCG2PDE4APDE4BPDE4CPDE4D
SCHEMBL9986622 0.86 ABCG2 (0.84) ABCG2PDE4APDE4BPDE4CPDE4D
SCHEMBL25191354 0.83 MAOB (0.77) ABCG2MEN1MAPTRAB9AKMT2A
SCHEMBL30382414 0.83 MAOB (0.77) ABCG2MEN1MAPTRAB9AKMT2A
SCHEMBL25195133 0.83 MAOB (0.77) ABCG2MEN1MAPTRAB9AKMT2A
SCHEMBL25204002 0.82 ABCG2 (0.68) ABCG2MEN1NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430047-A Neurotensin antagonists WARNER-LAMBERT COMPANY (US) 1995-07-04 US disclosed