SCHEMBL7333314

SCHEMBL7333314

c1ccc2nc(CCN3CCCCC3)ncc2c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.47
HRH3 Q9Y5N1 8/20 0.45
SLC6A3 Q01959 1/20 0.45
HTR3A P46098 1/20 0.43
HRH4 Q9H3N8 1/20 0.43
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP1A2 P05177 2/20 0.41
LTA4H P09960 1/20 0.41
KCNH2 Q12809 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
PARP1 P09874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1514879 0.85 SLC6A4 (0.50) SIGMAR1SLC6A3HTR3AHRH4MEN1
SCHEMBL1514937 0.81 FAAH (0.44) HRH4MEN1MAPTKMT2AKCNH2
SCHEMBL4965861 0.78 ACP1 (0.51) HRH3LTA4HKCNH2
SCHEMBL30117493 0.78 MEN1 (0.55) MEN1MAPTKMT2ACYP1A2LTA4H
SCHEMBL5649077 0.77 ACP1 (0.49) HRH3MEN1MAPTKMT2ALTA4H
SCHEMBL28184862 0.75 CYP1A2 (0.53) SIGMAR1HRH3SLC6A3CYP1A2CYP3A4
SCHEMBL5742502 0.74 KMT2A (0.47) MEN1MAPTKMT2A
SCHEMBL27269314 0.74 PDE10A (0.61) SIGMAR1HRH3SLC6A3MEN1MAPT
SCHEMBL460159 0.74 MAPK1 (0.41) HTR3AHRH4MEN1MAPTKMT2A
SCHEMBL28309633 0.73 HRH3 (0.53) SIGMAR1HRH3SLC6A3MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767792-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-11-20 EP disclosed
US-5977101-A Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity SMITHKLINE BEECHAM CORPORATION (US) 1999-11-02 US disclosed
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed
EP-0767792-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-04-16 EP disclosed
WO-1996000730-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1996-01-11 WO disclosed