SCHEMBL7333442

SCHEMBL7333442

COc1cccc(OC(C(=O)O)c2ccc3c(c2)OCO3)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.56
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
CTNNB1 P35222 1/20 0.53
WNT3A P56704 1/20 0.53
EDNRA P25101 3/20 0.53
MEN1 O00255 1/20 0.48
LMNA P02545 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
TP53 P04637 2/20 0.47
EDNRB P24530 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8791812 0.88 EDNRA (0.55) KMT2ANPC1RAB9AEDNRAALDH1A1
SCHEMBL2346146 0.81 KMT2A (0.56) KMT2AEDNRAMEN1ALDH1A1HPGD
SCHEMBL11402001 0.78 MEN1 (0.59) KMT2ANPC1RAB9AMEN1LMNA
SCHEMBL4824905 0.78 KMT2A (0.52) KMT2ANPC1RAB9ACTNNB1WNT3A
SCHEMBL6314113 0.75 KMT2A (0.45) KMT2AEDNRAMEN1ALDH1A1MAPT
SCHEMBL7329159 0.74 EDNRA (0.53) KMT2ANPC1RAB9AEDNRAALDH1A1
SCHEMBL27952103 0.73 KMT2A (0.71) KMT2AMEN1
SCHEMBL7331355 0.73 EDNRA (0.51) KMT2ACTNNB1WNT3AEDNRAMEN1
SCHEMBL27842527 0.73 KMT2A (0.54) KMT2ANPC1RAB9ACTNNB1WNT3A
SCHEMBL1580245 0.73 PTGS1 (0.65)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996009818-A1 ENDOTHELIN RECEPTOR ANTAGONISTS FOR THE TREATMENT OF EMESIS MERCK & CO., INC. (US) 1996-04-04 WO claimed
US-5767310-A Phenoxyphenylacetic acid derivatives MERCK & CO., INC. (US) 1998-06-16 US disclosed
US-5668176-A ENDOTHELIN ANTAGONIST MERCK & CO. INC. (US) 1997-09-16 US disclosed
US-5565485-A TREATING CARDIOVASCULAR DISORDERS MERCK & CO., INC. (US) 1996-10-15 US disclosed
WO-1996009818-A1 ENDOTHELIN RECEPTOR ANTAGONISTS FOR THE TREATMENT OF EMESIS MERCK & CO., INC. (US) 1996-04-04 WO disclosed
WO-1996004905-A1 PHENOXYPHENYLACETIC ACID DERIVATIVES MERCK & CO., INC. (US) 1996-02-22 WO disclosed
WO-1994021590-A1 PHENOXYPHENYLACETIC ACID DERIVATIVES MERCK & CO., INC. (US) 1994-09-29 WO disclosed
EP-0617001-A1 Phenoxyphenylacetic acid derivatives MERCK & CO. INC. (US) 1994-09-28 EP disclosed