SCHEMBL7334109

SCHEMBL7334109

N#Cc1ccc2cc(C(=O)Nc3ccc(N)cc3)ccc2c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 8/20 0.63
F2 P00734 3/20 0.63
PLG P00747 3/20 0.63
KLKB1 P03952 3/20 0.63
PRSS1 P07477 3/20 0.63
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
LMNA P02545 1/20 0.57
POLB P06746 1/20 0.57
PKM P14618 1/20 0.57
APEX1 P27695 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
ESR1 P03372 1/20 0.51
MLYCD O95822 1/20 0.50
TP53 P04637 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
DEGS1 O15121 1/20 0.50
SNCA P37840 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22695574 0.87 POLB (0.75) PLAUF2PLGKLKB1PRSS1
SCHEMBL7335211 0.86 PLAU (0.74) PLAUF2PLGKLKB1PRSS1
SCHEMBL7334216 0.85 PLAU (0.70) PLAUF2PLGKLKB1PRSS1
SCHEMBL20379456 0.85 MEN1 (0.73) PLAUF2PLGKLKB1PRSS1
SCHEMBL28013893 0.81 PLAU (0.74) PLAUF2PLGKLKB1PRSS1
SCHEMBL679200 0.81 DEGS1 (0.74) PLAUF2PLGKLKB1PRSS1
SCHEMBL7335241 0.77 PLAU (0.62) PLAUF2PLGKLKB1PRSS1
SCHEMBL28013896 0.77 PLAU (0.68) PLAUF2PLGKLKB1PRSS1
SCHEMBL5561129 0.77 PLAU (1.00) PLAUF2PLGKLKB1PRSS1
SCHEMBL9337665 0.77 MLYCD (0.76) PLAUF2PLGKLKB1PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284796-B1 NAPHTHAMIDINE COMPOUNDS ABBOTT LABORATORIES 2001-09-04 US disclosed
US-6258822-B1 ENZYME INHIBITORS OF NAPHTHALENE AMIDINE COMPOUNDS ABBOTT LABORATORIES 2001-07-10 US disclosed