SCHEMBL7335646

SCHEMBL7335646

CC(C)(C)[Si](C)(C)OCc1ccc(O)cc1OC(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.39
TRPV1 Q8NER1 3/20 0.33
TACR1 P25103 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
MAOB P27338 1/20 0.31
NTRK1 P04629 1/20 0.31
PDE2A O00408 1/20 0.31
APP P05067 1/20 0.30
RXRA P19793 1/20 0.30
RXRB P28702 1/20 0.30
RXRG P48443 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29375354 0.89 BACE1 (0.39) BACE1TRPV1TACR1FFAR4NTRK1
SCHEMBL26978999 0.89 BACE1 (0.39) BACE1TRPV1TACR1FFAR4NTRK1
SCHEMBL7334010 0.84 EPHX2 (0.40)
SCHEMBL23778772 0.79 BACE1 (0.41) BACE1
SCHEMBL29377447 0.77 CYP1A2 (0.33) BACE1TACR1NTRK1PDE2ARXRA
SCHEMBL26978199 0.77 CYP1A2 (0.33) BACE1TACR1NTRK1PDE2ARXRA
SCHEMBL30593420 0.76 GAA (0.38)
SCHEMBL2646502 0.76 CYP1A2 (0.34) BACE1PDE2A
SCHEMBL26979432 0.76 GAA (0.38)
SCHEMBL29377445 0.75 KCNH2 (0.33) BACE1TACR1NTRK1RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed
US-5968938-A Piperazine oxytocin receptor antagonists MERCK & CO., INC. (US) 1999-10-19 US disclosed