SCHEMBL7334010

SCHEMBL7334010

CC(C)(C)[Si](C)(C)OCc1ccc(Br)cc1OC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.40
ALPL P05186 6/20 0.39
ADRA2A P08913 5/20 0.36
MCHR1 Q99705 5/20 0.36
HRH4 Q9H3N8 2/20 0.35
NPY5R Q15761 2/20 0.35
SLC6A4 P31645 1/20 0.34
APLNR P35414 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26979432 0.89 GAA (0.38) EPHX2ALPLSLC6A4
SCHEMBL30593420 0.89 GAA (0.38) EPHX2ALPLSLC6A4
SCHEMBL7335646 0.84 BACE1 (0.39)
SCHEMBL29843138 0.84 PYCR1 (0.43)
SCHEMBL1430163 0.84 PYCR1 (0.43)
SCHEMBL24817103 0.84 HRH4 (0.39) EPHX2HRH4SLC6A4APLNR
SCHEMBL4513196 0.81 GAA (0.37) APLNR
SCHEMBL29771585 0.80 APLNR (0.43) APLNR
SCHEMBL1364662 0.80 APLNR (0.43) APLNR
SCHEMBL20512345 0.79 PYCR1 (0.36) APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090805-A Tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 2000-07-18 US disclosed
US-5968938-A Piperazine oxytocin receptor antagonists MERCK & CO., INC. (US) 1999-10-19 US disclosed