SCHEMBL7335693

SCHEMBL7335693

O=C(Nc1ccc(C(=O)N2CCc3cn[nH]c3-c3ccccc32)cn1)c1ccccc1-c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 11/20 0.53
AVPR1A P37288 9/20 0.49
OXTR P30559 1/20 0.49
AVPR1B P47901 2/20 0.45
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9059603 0.92 AVPR2 (0.51) AVPR2AVPR1AOXTRAVPR1BCHRNB2
SCHEMBL7319146 0.89 AVPR2 (0.48) AVPR2AVPR1AOXTRAVPR1BCHRNB2
SCHEMBL7333632 0.89 AVPR2 (0.64) AVPR2AVPR1AOXTRAVPR1B
SCHEMBL7337329 0.85 AVPR2 (0.46) AVPR2AVPR1A
SCHEMBL7335574 0.84 AVPR2 (0.61) AVPR2AVPR1A
SCHEMBL7339550 0.83 AVPR1A (0.51) AVPR2AVPR1AOXTRAVPR1B
SCHEMBL7337254 0.81 AVPR2 (0.52) AVPR2AVPR1AOXTR
SCHEMBL5945608 0.80 AVPR2 (0.49) AVPR2AVPR1AOXTRAVPR1BCHRNB2
SCHEMBL7342518 0.80 AVPR2 (0.80) AVPR2AVPR1A
SCHEMBL5237135 0.79 AVPR2 (0.54) AVPR2AVPR1AOXTRAVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO claimed
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed