SCHEMBL7337254

SCHEMBL7337254

O=C(c1ccc(-c2ccccc2)cc1)N1CCc2cn[nH]c2-c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 7/20 0.52
AVPR1A P37288 6/20 0.52
OXTR P30559 3/20 0.52
HPGD P15428 2/20 0.50
ALDH1A1 P00352 1/20 0.50
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
KMT2A Q03164 2/20 0.46
NPC1 O15118 1/20 0.46
ROCK2 O75116 1/20 0.45
STAT3 P40763 1/20 0.44
CYP11B2 P19099 1/20 0.43
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
MEN1 O00255 1/20 0.42
CRBN Q96SW2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8820724 0.89 AVPR2 (0.52) AVPR2AVPR1AHPGDALDH1A1RAB9A
SCHEMBL7333632 0.85 AVPR2 (0.64) AVPR2AVPR1AOXTR
SCHEMBL7335693 0.81 AVPR2 (0.53) AVPR2AVPR1AOXTR
SCHEMBL7332888 0.80 AVPR2 (0.65) AVPR2AVPR1AOXTRHPGDALDH1A1
SCHEMBL8820600 0.75 AVPR2 (0.53) AVPR2RAB9ASMN1; SMN2KMT2ANPC1
SCHEMBL7342518 0.74 AVPR2 (0.80) AVPR2AVPR1A
SCHEMBL7313684 0.73 AVPR2 (0.79) AVPR2AVPR1AOXTR
SCHEMBL9059603 0.73 AVPR2 (0.51) AVPR2AVPR1AOXTR
SCHEMBL5237135 0.73 AVPR2 (0.54) AVPR2AVPR1AOXTR
SCHEMBL2486302 0.73 HPGD (0.50) AVPR2AVPR1AHPGDALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed